SCHEMBL8091424

SCHEMBL8091424

CCOC(=O)C1=C(C)NC(C)=C(C(C)=O)C1c1ccccc1[N+](=O)[O-]

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1C Q13936 7/20 0.70
CACNA1D Q01668 7/20 0.70
CACNA1F O60840 5/20 0.70
CACNA1S Q13698 5/20 0.70
ADORA3 P0DMS8 5/20 0.70
ABCC4 O15439 2/20 0.70
ABCB11 O95342 2/20 0.70
LMNA P02545 2/20 0.70
CYP1A2 P05177 2/20 0.70
ADORA2A P29274 2/20 0.70
ADORA1 P30542 2/20 0.70
OPRM1 P35372 2/20 0.70
SCN1A P35498 2/20 0.70
HTR2B P41595 2/20 0.70
KCNH2 Q12809 2/20 0.70
SCN5A Q14524 2/20 0.70
SCN2A Q99250 2/20 0.70
SCN3A Q9NY46 2/20 0.70
CACNA1B Q00975 2/20 0.70
MAPT P10636 2/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29810716 0.95 CACNA1C (0.77) CACNA1CCACNA1DCACNA1FCACNA1SADORA3
SCHEMBL1617472 0.95 CACNA1C (0.77) CACNA1CCACNA1DCACNA1FCACNA1SADORA3
SCHEMBL5085498 0.91 ADORA3 (0.86) CACNA1CCACNA1DCACNA1FCACNA1SADORA3
SCHEMBL7266381 0.91 CACNA1B (0.74) CACNA1CCACNA1DCACNA1FCACNA1SADORA3
SCHEMBL7412221 0.91 CACNA1B (0.74) CACNA1CCACNA1DCACNA1FCACNA1SADORA3
SCHEMBL29358809 0.89 CACNA1C (0.73) CACNA1CCACNA1DCACNA1FCACNA1SADORA3
SCHEMBL202183 0.89 CACNA1C (0.73) CACNA1CCACNA1DCACNA1FCACNA1SADORA3
SCHEMBL11524993 0.88 CACNA1C (0.67) CACNA1CCACNA1DCACNA1FCACNA1SADORA3
SCHEMBL8048696 0.88 ADORA3 (0.90) CACNA1CCACNA1DCACNA1FCACNA1SADORA3
SCHEMBL9765770 0.88 CACNA1C (0.86) CACNA1CCACNA1DCACNA1FCACNA1SADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3966948-A Spasmolytic, vaso-dilating and anti-hypertensive compositions and methods BAYER AKTIENGESELLSCHAFT (DT) 1976-06-29 US claimed
US-6067135-A Liquid crystal display device and method of manufacturing the same KABUSHIKI KAISHA TOSHIBA (JP) 2000-05-23 US disclosed
US-4593100-A 3A,4,7,7a-tetrahydro-3,6,7a-trimethyl-4-substituted phenyl-isoxazolo[5,4-b]pyridine-5-carboxylic acid esters AMERICAN HOME PRODUCTS CORPORATION (US) 1986-06-03 US disclosed
US-3966948-A Spasmolytic, vaso-dilating and anti-hypertensive compositions and methods BAYER AKTIENGESELLSCHAFT (DT) 1976-06-29 US disclosed