SCHEMBL8091845

SCHEMBL8091845

C[C@@H](CO)NC(=O)Nc1ccc(-c2nc(N)cc(C3(S(=O)(=O)c4ccc(F)cc4)CCC3)n2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 3/20 0.38
MTOR P42345 2/20 0.38
ALDH1A1 P00352 1/20 0.38
CA2 P00918 4/20 0.37
CA9 Q16790 4/20 0.37
CA12 O43570 3/20 0.37
CA1 P00915 3/20 0.37
RORC P51449 2/20 0.36
NAMPT P43490 1/20 0.36
FPR2 P25090 1/20 0.36
SCN9A Q15858 1/20 0.36
RAB9A P51151 1/20 0.35
KDM1A O60341 1/20 0.34
CA4 P22748 1/20 0.34
CA7 P43166 1/20 0.34
PIK3CG P48736 1/20 0.34
KMT2A Q03164 1/20 0.34
PIK3CD O00329 3/20 0.34
CYP2C9 P11712 1/20 0.34
IDO1 P14902 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8092462 1.00 PIK3CA (0.38) PIK3CAMTORALDH1A1CA2CA9
SCHEMBL8098658 0.92 MAPT (0.37) PIK3CAALDH1A1CA2CA9CA12
SCHEMBL8098657 0.92 MAPT (0.37) PIK3CAALDH1A1CA2CA9CA12
SCHEMBL8097581 0.88 MAPT (0.38) PIK3CAALDH1A1CA2CA9CA12
SCHEMBL8091937 0.87 CA12 (0.39) PIK3CAMTORALDH1A1CA2CA9
SCHEMBL8100146 0.86 CA1 (0.41) PIK3CAMTORALDH1A1CA2CA9
SCHEMBL8093158 0.85 PIK3CA (0.38) PIK3CAMTORALDH1A1CA2CA9
SCHEMBL8084990 0.85 CA1 (0.40) PIK3CAMTORALDH1A1CA2CA9
SCHEMBL8097426 0.84 NAMPT (0.41) PIK3CAMTORALDH1A1CA2CA9
SCHEMBL8089094 0.84 PIK3CD (0.43) PIK3CAMTORALDH1A1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed