SCHEMBL8092836

SCHEMBL8092836

Oc1ccc(CCCNCCCc2ccccc2)cc1

nearest known ligand 0.93

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 8/20 0.76
MPO P05164 1/20 0.59
DRD2 P14416 1/20 0.58
DRD4 P21917 1/20 0.58
DRD3 P35462 1/20 0.58
KCNH2 Q12809 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12009648 0.96 SIGMAR1 (0.78) SIGMAR1DRD3KCNH2
SCHEMBL3866233 0.91 SIGMAR1 (0.70) SIGMAR1MPO
SCHEMBL3692847 0.91 SIGMAR1 (0.70) SIGMAR1MPO
SCHEMBL7379499 0.91 SIGMAR1 (0.79) SIGMAR1DRD3KCNH2
SCHEMBL18122725 0.88 OPRK1 (0.64) SIGMAR1MPODRD3KCNH2
SCHEMBL4254894 0.87 SIGMAR1 (1.00) SIGMAR1DRD2DRD4DRD3KCNH2
Methyl Alcohol SCHEMBL7281789 0.85 SIGMAR1 (0.68) SIGMAR1DRD3KCNH2
SCHEMBL2538905 0.85 SIGMAR1 (0.95) SIGMAR1DRD2DRD4DRD3KCNH2
SCHEMBL157572 0.85 DPP4 (0.63)
SCHEMBL1238323 0.85 ESR1 (0.62) SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057371-A TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS, GASTROINTESTINAL DISORDERS, DRUG ABUSE, ANGINA, MIGRAINE, HYPERTENSION AND DEPRESSION VIRGINIA COMMONWEALTH UNIVERSITY (US) 2000-05-02 US disclosed
EP-0591426-A1 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1994-04-13 EP disclosed
EP-0507863-A4 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF 1993-07-07 EP disclosed
WO-1993000313-A2 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1993-01-07 WO disclosed
EP-0507863-A1 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1992-10-14 EP disclosed
WO-1991009594-A1 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1991-07-11 WO disclosed