SCHEMBL8093490

SCHEMBL8093490

N#Cc1cc(-c2ccc(S(N)(=O)=O)cc2)c(-c2ccc(F)cc2)nc1SCC(=O)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.51
LMNA P02545 2/20 0.51
CA2 P00918 11/20 0.50
CA9 Q16790 10/20 0.50
CA1 P00915 10/20 0.50
CA12 O43570 9/20 0.50
CA7 P43166 2/20 0.45
CA13 Q8N1Q1 2/20 0.45
MAPT P10636 5/20 0.45
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
USP2 O75604 2/20 0.45
NPSR1 Q6W5P4 2/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
CA4 P22748 1/20 0.44
RECQL P46063 1/20 0.44
ALOX15 P16050 1/20 0.44
MAPK1 P28482 1/20 0.44
HSD17B10 Q99714 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8101120 0.91 ALDH1A1 (0.51) ALDH1A1LMNACA2CA9CA1
SCHEMBL8093715 0.84 CNR1 (0.46) ALDH1A1CA2CA9CA1CA12
SCHEMBL8095872 0.83 ALDH1A1 (0.55) ALDH1A1LMNAMAPTMEN1KMT2A
SCHEMBL8093864 0.83 CA9 (0.44) CA2CA9CA1CA12CA4
SCHEMBL8094384 0.82 MAPK13 (0.47) ALDH1A1LMNACA2CA9CA1
SCHEMBL8104361 0.80 ALDH1A1 (0.46) ALDH1A1LMNACA2CA9CA1
SCHEMBL8093245 0.80 ALDH1A1 (0.45) ALDH1A1LMNACA2CA9CA1
SCHEMBL8423226 0.80 ALDH1A1 (0.48) ALDH1A1LMNACA2CA9CA1
SCHEMBL8095741 0.79 PDE10A (0.43) ALDH1A1LMNACA2CA9CA1
SCHEMBL8086490 0.78 ALDH1A1 (0.42) ALDH1A1LMNACA2CA9CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808304-B1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2000-12-27 EP disclosed
EP-0808304-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1997-11-26 EP disclosed
WO-1996024584-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-08-15 WO disclosed