SCHEMBL8093864

SCHEMBL8093864

N#Cc1cc(-c2ccc(S(N)(=O)=O)cc2)c(-c2ccc(F)cc2)nc1NCC(=O)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 10/20 0.44
CA1 P00915 9/20 0.44
CA2 P00918 9/20 0.44
CA12 O43570 8/20 0.44
PTGS2 P35354 6/20 0.42
PTGS1 P23219 3/20 0.41
CA4 P22748 2/20 0.39
CDK1 P06493 1/20 0.38
KDR P35968 1/20 0.38
CHRNA7 P36544 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8099443 0.91 PTGS2 (0.50) PTGS2PTGS1
SCHEMBL8093715 0.85 CNR1 (0.46) CA9CA1CA2CA12PTGS2
SCHEMBL8094849 0.84 HPGD (0.48) CA9CA1CA2CA12PTGS2
SCHEMBL8092670 0.83 GLA (0.44) CA9CA1CA2CA12PTGS2
SCHEMBL8093490 0.83 ALDH1A1 (0.51) CA9CA1CA2CA12CA4
SCHEMBL8092536 0.82 PTGS2 (0.43) CA9CA1CA2CA12PTGS2
SCHEMBL8421223 0.81 NPSR1 (0.41)
SCHEMBL8086911 0.81 HPGD (0.45) CA9CA1CA2CA12PTGS2
SCHEMBL8093987 0.80 PTGS2 (0.48) CA9CA1CA2CA12PTGS2
SCHEMBL8094187 0.79 CNR1 (0.50) CA9CA1CA2CA12PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808304-B1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2000-12-27 EP disclosed