SCHEMBL8093527

SCHEMBL8093527

Cc1ccc(Nc2nc(-c3ccc(Cl)cc3)nc3ccccc23)cc1

nearest known ligand 0.82

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 9/20 0.82
MAPT P10636 5/20 0.82
TP53 P04637 3/20 0.82
PDE5A O76074 3/20 0.82
LMNA P02545 1/20 0.82
MEN1 O00255 4/20 0.77
KMT2A Q03164 4/20 0.77
GAA P10253 2/20 0.77
GBA1 P04062 1/20 0.77
POLB P06746 1/20 0.77
KDM4E B2RXH2 1/20 0.74
ALDH1A1 P00352 1/20 0.74
RXFP1 Q9HBX9 1/20 0.74
MAPK1 P28482 2/20 0.66
HTT P42858 1/20 0.66
NPSR1 Q6W5P4 1/20 0.65
NTSR1 P30989 1/20 0.65
KDM1A O60341 2/20 0.62
ALK Q9UM73 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22201364 0.93 ABCG2 (0.94) ABCG2MAPTTP53PDE5ALMNA
SCHEMBL8095812 0.90 ABCG2 (1.00) ABCG2MAPTTP53PDE5ALMNA
SCHEMBL5531993 0.90 ABCG2 (0.89) ABCG2MAPTTP53PDE5ALMNA
SCHEMBL4867505 0.90 ABCG2 (1.00) ABCG2MAPTTP53PDE5ALMNA
SCHEMBL12316824 0.87 GAA (1.00) ABCG2MAPTTP53PDE5ALMNA
SCHEMBL8096433 0.86 ABCG2 (0.83) ABCG2MAPTTP53PDE5ALMNA
SCHEMBL1064901 0.85 TGFBR1 (0.82) ABCG2MAPTTP53PDE5ALMNA
SCHEMBL1083796 0.85 KDM4E (1.00) ABCG2MAPTTP53PDE5ALMNA
SCHEMBL13945460 0.85 ABCG2 (0.83) ABCG2MAPTTP53PDE5ALMNA
SCHEMBL8087337 0.85 ABCG2 (0.85) ABCG2MAPTTP53PDE5ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009000085-A1 QUINOLINE AND QUINAZOLINE DERIVATIVES USEFUL AS MODULATORS OF GATED ION CHANNELS PAINCEPTOR PHARMA CORPORATION (CA) 2008-12-31 WO disclosed