SCHEMBL8093579

SCHEMBL8093579

CC(=O)c1ccc(N=C=O)cc1.CC(C)c1ccc(N=C=O)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.46
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
NOS3 P29474 2/20 0.44
NOS1 P29475 2/20 0.44
MAPK1 P28482 4/20 0.43
SMN1; SMN2 Q16637 4/20 0.43
TDP1 Q9NUW8 2/20 0.43
STAT3 P40763 1/20 0.43
STAT1 P42224 1/20 0.43
PRSS1 P07477 1/20 0.41
ACR P10323 1/20 0.41
CYP2C9 P11712 2/20 0.41
SCN5A Q14524 1/20 0.40
SCN2A Q99250 1/20 0.40
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40
USP5 P45974 1/20 0.40
TP53 P04637 1/20 0.40
THRB P10828 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL219763 0.88 NOS3 (0.55) MAPTNPC1RAB9ANOS3NOS1
SCHEMBL131853 0.86 CYP3A4 (0.50) MAPTNPC1RAB9ANOS3NOS1
SCHEMBL182327 0.82 CYP2C9 (0.55) MAPTNPC1RAB9ANOS3NOS1
Hydrochloric Acid SCHEMBL5197216 0.80 CYP2C9 (0.53) MAPTNPC1RAB9ANOS3NOS1
SCHEMBL7005068 0.79 CYP3A4 (0.44) MAPTRAB9AMAPK1SMN1; SMN2TDP1
SCHEMBL13851927 0.78 TSHR (0.69) MAPTNPC1RAB9ANOS3NOS1
SCHEMBL8724560 0.77 HPGD (0.48) MAPTNPC1RAB9ANOS3NOS1
SCHEMBL12591838 0.76 SMN1; SMN2 (0.59) MAPTRAB9AMAPK1SMN1; SMN2CYP2C9
SCHEMBL21934213 0.76 CYP3A4 (0.71) NOS3NOS1MAPK1SMN1; SMN2TDP1
SCHEMBL27705454 0.75 CYP3A4 (0.44) MAPK1TDP1CYP2C9CYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973936-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC AMINOTHIOETHER ACIDS ELI LILLY AND COMPANY (US) 2000-01-26 EP disclosed
WO-1998046786-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC AMINOTHIOETHER ACIDS ELI LILLY AND COMPANY (US) 1998-10-22 WO disclosed