SCHEMBL8094067

SCHEMBL8094067

CNc1nc(-c2ccc(F)cc2)c(-c2ccc(S(C)(=O)=O)cc2)cc1C#N

nearest known ligand 0.49

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 19/20 0.49
PTGS1 P23219 2/20 0.48
CNR1 P21554 1/20 0.45
CNR2 P34972 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8776825 0.89 PTGS2 (0.46) PTGS2PTGS1CNR1CNR2
SCHEMBL8095222 0.86 PTGS2 (0.53) PTGS2PTGS1
SCHEMBL8098348 0.85 PTGS2 (0.52) PTGS2PTGS1
SCHEMBL8098107 0.85 PTGS2 (0.52) PTGS2PTGS1
SCHEMBL8095119 0.84 HPGD (0.47) PTGS2PTGS1
SCHEMBL212410 0.84 PTGS2 (0.51) PTGS2PTGS1
SCHEMBL8087025 0.84 PTGS2 (0.54) PTGS2PTGS1
SCHEMBL8099266 0.84 PTGS2 (0.53) PTGS2PTGS1
SCHEMBL8101771 0.83 PTGS2 (0.54) PTGS2PTGS1CNR1CNR2
SCHEMBL8093654 0.83 PTGS2 (0.50) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808304-B1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2000-12-27 EP claimed
EP-0808304-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1997-11-26 EP claimed
WO-1996024584-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-08-15 WO claimed
EP-0808304-B1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2000-12-27 EP disclosed
US-5916905-A ANTIARTHRITIC AGENTS; ANALGESICS; ANTIPYRETICS G. D. SEARLE & CO. (US) 1999-06-29 US disclosed
US-5686470-A 2, 3-substituted pyridines for the treatment of inflammation WEIER RICHARD M (US) 1997-11-11 US disclosed