SCHEMBL8776825

SCHEMBL8776825

CCS(=O)(=O)c1ccc(-c2cc(C#N)c(NC)nc2-c2ccc(F)cc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 9/20 0.46
CNR1 P21554 4/20 0.44
CNR2 P34972 1/20 0.44
RORC P51449 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
GAA P10253 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
PTGS1 P23219 2/20 0.40
AKT1 P31749 1/20 0.40
AKT2 P31751 1/20 0.40
SCN9A Q15858 2/20 0.38
ADORA1 P30542 1/20 0.38
ERBB2 P04626 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8094067 0.89 PTGS2 (0.49) PTGS2CNR1CNR2PTGS1
SCHEMBL8776749 0.84 PTGS2 (0.47) PTGS2CNR1CNR2RORCALDH1A1
SCHEMBL8776720 0.83 PTGS2 (0.47) PTGS2CNR1CNR2KDM4EPTGS1
SCHEMBL8776822 0.80 PTGS2 (0.56) PTGS2CNR1CNR2PTGS1SCN9A
SCHEMBL8776765 0.77 CNR1 (0.60) PTGS2CNR1CNR2KDM4EPTGS1
SCHEMBL8095119 0.76 HPGD (0.47) PTGS2KDM4EALDH1A1PTGS1
SCHEMBL8776719 0.76 PTGS2 (0.44) PTGS2CNR1CNR2RORCKDM4E
SCHEMBL8099266 0.76 PTGS2 (0.53) PTGS2ALDH1A1SMN1; SMN2PTGS1
SCHEMBL8100740 0.75 PTGS2 (0.58) PTGS2CNR1PTGS1
SCHEMBL8101771 0.75 PTGS2 (0.54) PTGS2CNR1CNR2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808304-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1997-11-26 EP disclosed
WO-1996024584-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-08-15 WO disclosed