SCHEMBL8094130

SCHEMBL8094130

O=S(=O)(c1cccs1)N1CC(CN2CCC(c3ccccc3)CC2)C(c2ccccc2)C1

nearest known ligand 0.74

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 19/20 0.74
MEN1 O00255 1/20 0.48
ALDH1A1 P00352 1/20 0.48
POLB P06746 1/20 0.48
TSHR P16473 1/20 0.48
MAPK1 P28482 1/20 0.48
KMT2A Q03164 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7836739 0.84 CCR5 (1.00) CCR5
SCHEMBL7835509 0.81 CCR5 (0.87) CCR5
SCHEMBL7817814 0.80 CCR5 (0.85) CCR5
SCHEMBL7826200 0.78 CCR5 (0.78) CCR5ALDH1A1
SCHEMBL7836855 0.78 CCR5 (0.71) CCR5
SCHEMBL7833942 0.74 CCR5 (1.00) CCR5
SCHEMBL7825773 0.74 CCR5 (0.65) CCR5MEN1ALDH1A1TSHRMAPK1
SCHEMBL7836524 0.70 CCR5 (1.00) CCR5MEN1TSHRKMT2A
SCHEMBL5174991 0.70 CCR5 (0.74) CCR5MEN1KMT2A
SCHEMBL8090790 0.69 CCR5 (1.00) CCR5MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6166037-A Pyrrolidine and piperidine modulators of chemokine receptor activity MERCK & CO., INC. (US) 2000-12-26 US disclosed