SCHEMBL8094187

SCHEMBL8094187

N#Cc1cc(-c2ccc(S(N)(=O)=O)cc2)c(-c2ccc(F)cc2)nc1NCc1ccc(Cl)cc1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 10/20 0.50
CNR2 P34972 5/20 0.50
CA1 P00915 3/20 0.46
CA2 P00918 3/20 0.46
CA7 P43166 1/20 0.46
CA13 Q8N1Q1 1/20 0.46
MAP3K8 P41279 1/20 0.44
PTGS2 P35354 3/20 0.43
CA12 O43570 2/20 0.42
CA9 Q16790 2/20 0.42
CA14 Q9ULX7 1/20 0.42
MALT1 Q9UDY8 1/20 0.42
CDK1 P06493 1/20 0.42
KDR P35968 1/20 0.42
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8101771 0.91 PTGS2 (0.54) CNR1CNR2PTGS2
SCHEMBL8093987 0.90 PTGS2 (0.48) CNR1CNR2CA1CA2CA7
SCHEMBL8085724 0.86 PTGS2 (0.51) CNR1CNR2CA1CA2CA7
SCHEMBL8095797 0.84 CNR1 (0.69) CNR1CNR2CA1CA2CA7
SCHEMBL8092536 0.84 PTGS2 (0.43) CNR1CNR2CA1CA2CA13
SCHEMBL8086911 0.83 HPGD (0.45) CNR1CNR2CA1CA2PTGS2
SCHEMBL8086615 0.83 PTGS2 (0.49) CNR1CNR2CA1CA2PTGS2
SCHEMBL8099660 0.82 MAPT (0.49) CNR1CA1CA2CA7PTGS2
SCHEMBL8094849 0.82 HPGD (0.48) CA1CA2CA7CA13PTGS2
SCHEMBL8099266 0.80 PTGS2 (0.53) PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808304-B1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2000-12-27 EP disclosed
EP-0808304-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1997-11-26 EP disclosed
WO-1996024584-A1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-08-15 WO disclosed