SCHEMBL8095797

SCHEMBL8095797

N#Cc1cc(-c2ccc(S(N)(=O)=O)cc2)c(-c2ccc(F)cc2)nc1OCc1ccc(Cl)cc1

nearest known ligand 0.69

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 17/20 0.69
CNR2 P34972 4/20 0.58
PTGS1 P23219 1/20 0.45
PTGS2 P35354 1/20 0.45
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA7 P43166 1/20 0.45
CA9 Q16790 1/20 0.45
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8086461 0.95 CNR1 (0.61) CNR1CNR2PTGS1PTGS2CA12
SCHEMBL8086096 0.91 CNR1 (0.69) CNR1CNR2PTGS1PTGS2
SCHEMBL8093875 0.91 CNR1 (0.64) CNR1CNR2PTGS1PTGS2CA12
SCHEMBL8093740 0.89 CNR1 (0.60) CNR1CNR2PTGS1PTGS2CA12
SCHEMBL8095103 0.85 CNR1 (0.61) CNR1CNR2PTGS1PTGS2
SCHEMBL8094678 0.85 SQOR (0.53) CNR1CNR2PTGS2ALDH1A1
SCHEMBL8094551 0.84 CNR1 (0.49) CNR1CNR2PTGS1PTGS2CA12
SCHEMBL8094187 0.84 CNR1 (0.50) CNR1CNR2PTGS2CA12CA1
SCHEMBL8101417 0.83 CNR1 (0.50) CNR1CNR2PTGS1PTGS2CA12
SCHEMBL8095521 0.82 CNR1 (0.52) CNR1PTGS1PTGS2CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808304-B1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2000-12-27 EP claimed
EP-0808304-B1 2,3-SUBSTITUTED PYRIDINES FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2000-12-27 EP disclosed