SCHEMBL8094473

SCHEMBL8094473

Cc1cc([N+](=O)[O-])cc(C)c1C(=O)Br

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.52
GPR35 Q9HC97 1/20 0.52
TDP1 Q9NUW8 3/20 0.50
CYP3A4 P08684 3/20 0.50
TSHR P16473 3/20 0.48
HTT P42858 3/20 0.44
KMT2A Q03164 3/20 0.44
MEN1 O00255 2/20 0.44
LMNA P02545 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.42
MAPT P10636 1/20 0.42
CYP19A1 P11511 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
L3MBTL1 Q9Y468 3/20 0.40
GALR3 O60755 1/20 0.40
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16632905 0.82 ALDH1A1 (0.53) ALDH1A1GPR35TDP1CYP3A4TSHR
SCHEMBL13199182 0.82 CA1 (0.55) ALDH1A1GPR35TDP1CYP3A4TSHR
SCHEMBL8099774 0.80 ALDH1A1 (0.52) ALDH1A1GPR35TDP1CYP3A4TSHR
SCHEMBL16633153 0.79 GSK3B (0.51) ALDH1A1GPR35TDP1CYP3A4TSHR
SCHEMBL14892423 0.78 ALDH1A1 (0.50) ALDH1A1GPR35TDP1CYP3A4TSHR
SCHEMBL27484194 0.77 MEN1 (0.50) ALDH1A1GPR35TDP1CYP3A4TSHR
SCHEMBL7591817 0.76 ALDH1A1 (0.49) ALDH1A1GPR35TDP1CYP3A4TSHR
SCHEMBL11980144 0.76 CA1 (0.67) ALDH1A1GPR35TDP1CYP3A4TSHR
SCHEMBL1286515 0.76 CA1 (0.67) ALDH1A1GPR35TDP1CYP3A4TSHR
SCHEMBL8101943 0.76 ALDH1A1 (0.59) ALDH1A1TDP1CYP3A4TSHRHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0708077-B1 Diamino compounds and methods for preparing them CHISSO CORP (JP) 2000-12-27 EP disclosed
US-5663440-A Diamino compounds and methods for preparing them CHISSO CORPORATION (JP) 1997-09-02 US disclosed
EP-0708077-A1 Diamino compounds and methods for preparing them CHISSO CORPORATION (JP) 1996-04-24 EP disclosed