SCHEMBL8094950

SCHEMBL8094950

CCCc1cccc(C(=O)Cl)c1C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
ALOX15 P16050 1/20 0.37
MRGPRX4 Q96LA9 1/20 0.37
GABRA1 P14867 1/20 0.36
GABRB2 P47870 1/20 0.36
DAO P14920 1/20 0.36
TSHR P16473 1/20 0.36
HCRTR1 O43613 2/20 0.36
HCRTR2 O43614 2/20 0.36
IAPP P10997 1/20 0.36
HTT P42858 2/20 0.35
CYP1A2 P05177 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2D6 P10635 2/20 0.35
CYP2C19 P33261 2/20 0.35
CYP2C9 P11712 1/20 0.35
CLCN2 P51788 1/20 0.35
PPARG P37231 1/20 0.35
PPARA Q07869 1/20 0.35
TP53 P04637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8095512 0.90 BID (0.42) ALOX15TSHRIAPPHTTCYP3A4
SCHEMBL8087557 0.88 BID (0.48) ALOX15PPARGPPARABIDBCL2L1
SCHEMBL1892417 0.87 GABRA1 (0.45) ALDH1A1ALOX15MRGPRX4GABRA1GABRB2
SCHEMBL8094232 0.87 BID (0.50) ALOX15PPARGPPARABIDBCL2L1
SCHEMBL8093905 0.87 BID (0.50) ALOX15PPARGPPARABIDBCL2L1
SCHEMBL8095850 0.87 BID (0.50) ALOX15PPARGPPARABIDBCL2L1
SCHEMBL28642784 0.85 GABRA1 (0.39) ALDH1A1GABRA1GABRB2DAOTSHR
SCHEMBL2362450 0.84 MRGPRX4 (0.47) ALDH1A1ALOX15MRGPRX4TSHRHTT
SCHEMBL22620361 0.84 PRKCI (0.42) ALDH1A1GABRA1GABRB2DAOTSHR
SCHEMBL3180114 0.83 ALDH1A1 (0.45) ALDH1A1ALOX15TSHRHCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016044390-A1 BORON-CONTAINING DIACYLHYDRAZINE COMPOUNDS INTREXON CORPORATION (US) 2016-03-24 WO disclosed
EP-0708077-B1 Diamino compounds and methods for preparing them CHISSO CORP (JP) 2000-12-27 EP disclosed
US-5663440-A Diamino compounds and methods for preparing them CHISSO CORPORATION (JP) 1997-09-02 US disclosed
EP-0708077-A1 Diamino compounds and methods for preparing them CHISSO CORPORATION (JP) 1996-04-24 EP disclosed