SCHEMBL8095358

SCHEMBL8095358

CC(=O)NC[C@@H]1C[C@H]1c1cccc(Br)c1

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 3/20 0.55
HTR2A P28223 1/20 0.55
HTR2B P41595 1/20 0.55
KDM1A O60341 2/20 0.46
MTNR1A P48039 7/20 0.46
MTNR1B P49286 7/20 0.46
SLC6A4 P31645 2/20 0.43
SLC6A3 Q01959 1/20 0.43
CNR1 P21554 1/20 0.42
F2RL1 P55085 1/20 0.40
HDAC4 P56524 1/20 0.40
HRH3 Q9Y5N1 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8095359 1.00 HTR2C (0.55) HTR2CHTR2AHTR2BKDM1AMTNR1A
SCHEMBL8104287 0.86 HTR2C (0.52) HTR2CHTR2AHTR2BKDM1AMTNR1A
SCHEMBL8104288 0.86 HTR2C (0.52) HTR2CHTR2AHTR2BKDM1AMTNR1A
SCHEMBL8098498 0.84 HTR2C (0.56) HTR2CHTR2AHTR2BMTNR1AMTNR1B
SCHEMBL8098497 0.84 HTR2C (0.56) HTR2CHTR2AHTR2BMTNR1AMTNR1B
SCHEMBL8098175 0.84 MTNR1B (0.51) HTR2CHTR2AHTR2BKDM1AMTNR1A
SCHEMBL8098179 0.84 MTNR1B (0.51) HTR2CHTR2AHTR2BKDM1AMTNR1A
SCHEMBL8102597 0.83 HTR2C (0.56) HTR2CHTR2AHTR2BMTNR1AMTNR1B
SCHEMBL8102591 0.83 HTR2C (0.56) HTR2CHTR2AHTR2BMTNR1AMTNR1B
SCHEMBL4126434 0.82 HTR2A (0.51) HTR2CHTR2AHTR2BKDM1ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0747346-B1 N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL MYERS SQUIBB CO (US) 2000-02-16 EP disclosed
EP-0747346-A2 N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL-MYERS SQUIBB COMPANY (US) 1996-12-11 EP disclosed