SCHEMBL8104288

SCHEMBL8104288

CCC(=O)NCC1CC1c1cccc(Br)c1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.52
HTR2A P28223 1/20 0.52
HTR2B P41595 1/20 0.52
MTNR1B P49286 11/20 0.52
MTNR1A P48039 10/20 0.49
GAA P10253 1/20 0.47
KDM1A O60341 2/20 0.44
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.41
CNR1 P21554 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8104287 1.00 HTR2C (0.52) HTR2CHTR2AHTR2BMTNR1BMTNR1A
SCHEMBL8098179 0.90 MTNR1B (0.51) HTR2CHTR2AHTR2BMTNR1BMTNR1A
SCHEMBL8098175 0.90 MTNR1B (0.51) HTR2CHTR2AHTR2BMTNR1BMTNR1A
SCHEMBL8095359 0.86 HTR2C (0.55) HTR2CHTR2AHTR2BMTNR1BMTNR1A
SCHEMBL8095358 0.86 HTR2C (0.55) HTR2CHTR2AHTR2BMTNR1BMTNR1A
SCHEMBL8098094 0.84 HTR2C (0.54) HTR2CHTR2AHTR2BMTNR1BMTNR1A
SCHEMBL8098093 0.84 HTR2C (0.54) HTR2CHTR2AHTR2BMTNR1BMTNR1A
SCHEMBL8095717 0.82 HTR2A (0.58) HTR2CHTR2AHTR2BMTNR1BMTNR1A
SCHEMBL8095719 0.82 HTR2A (0.58) HTR2CHTR2AHTR2BMTNR1BMTNR1A
SCHEMBL4126434 0.80 HTR2A (0.51) HTR2CHTR2AHTR2BKDM1ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0747346-B1 N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL MYERS SQUIBB CO (US) 2000-02-16 EP disclosed
EP-0747346-A2 N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL-MYERS SQUIBB COMPANY (US) 1996-12-11 EP disclosed