SCHEMBL8095790

SCHEMBL8095790

O=C(NC[C@@H]1C[C@H]1c1cc(F)ccc1F)C1CC1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 6/20 0.47
MTNR1B P49286 6/20 0.47
HTR2A P28223 7/20 0.44
KDM1A O60341 2/20 0.44
KDM1B Q8NB78 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.43
HTR2C P28335 7/20 0.43
HTR2B P41595 4/20 0.43
FFAR1 O14842 1/20 0.41
GAA P10253 1/20 0.39
RIPK1 Q13546 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8089388 0.84 MTNR1B (0.52) MTNR1AMTNR1BHTR2AKDM1AKDM1B
SCHEMBL8089391 0.84 MTNR1B (0.52) MTNR1AMTNR1BHTR2AKDM1AKDM1B
SCHEMBL8104739 0.84 HTR2A (0.47) MTNR1AMTNR1BHTR2AKDM1AKDM1B
SCHEMBL8104735 0.84 HTR2A (0.47) MTNR1AMTNR1BHTR2AKDM1AKDM1B
SCHEMBL8097747 0.80 MTNR1B (0.51) MTNR1AMTNR1BHTR2AKDM1AKDM1B
SCHEMBL8097743 0.80 MTNR1B (0.51) MTNR1AMTNR1BHTR2AKDM1AKDM1B
SCHEMBL16585430 0.74 KDM1A (0.58) HTR2AKDM1AKDM1BHTR2CHTR2B
SCHEMBL17985315 0.74 KDM1A (0.58) HTR2AKDM1AKDM1BHTR2CHTR2B
SCHEMBL706719 0.74 KDM1A (0.58) HTR2AKDM1AKDM1BHTR2CHTR2B
SCHEMBL17962670 0.73 HTR2C (0.44) HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0747346-B1 N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL MYERS SQUIBB CO (US) 2000-02-16 EP disclosed
EP-0747346-A2 N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL-MYERS SQUIBB COMPANY (US) 1996-12-11 EP disclosed