SCHEMBL8095955

SCHEMBL8095955

C#Cc1ccc(-n2cnc(C)c2)c(N)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR2E1 Q9Y466 1/20 0.37
MAP3K14 Q99558 1/20 0.36
PSEN1 P49768 9/20 0.36
PSEN2 P49810 9/20 0.36
APH1B Q8WW43 9/20 0.36
NCSTN Q92542 9/20 0.36
APH1A Q96BI3 9/20 0.36
PSENEN Q9NZ42 9/20 0.36
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP19A1 P11511 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
CYP2E1 P05181 1/20 0.35
CYP2A6 P11509 1/20 0.35
GABRG2 P18507 2/20 0.34
GABRB3 P28472 2/20 0.34
GABRA5 P31644 2/20 0.34
KCNH2 Q12809 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3056259 0.82 USP30 (0.41) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL3040146 0.80 PSEN1 (0.41) NR2E1PSEN1PSEN2APH1BNCSTN
SCHEMBL3045214 0.80 PSEN1 (0.52) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL3056041 0.75 PSEN1 (0.41) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL3040182 0.74 CYP1A2 (0.55) NR2E1CYP1A2CYP3A4CYP2D6CYP19A1
SCHEMBL3055463 0.74 PSEN1 (0.43) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL27819262 0.73 GAA (0.48) NR2E1PSEN1PSEN2APH1BNCSTN
SCHEMBL3050264 0.71 CYP2E1 (0.41) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL1616168 0.70 ALDH1A1 (0.49) NR2E1PSEN1PSEN2APH1BNCSTN
SCHEMBL23119173 0.68 LMNA (0.41) NR2E1PSEN1PSEN2APH1BNCSTN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008156580-A1 TRIAZOLE DERIVATIVES FOR TREATING ALZHEIMER'S DISEASE AND RELATED CONDITIONS MERCK & CO., INC. (US) 2008-12-24 WO disclosed