SCHEMBL8097344

SCHEMBL8097344

N#Cc1ccc(Cc2cnc(Cc3ccc(-c4ccc(F)cc4Cl)cc3)[nH]2)cc1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BRS3 P32247 8/20 0.50
GCGR P47871 1/20 0.39
MAPK14 Q16539 1/20 0.39
CYP11B1 P15538 2/20 0.38
CYP11B2 P19099 2/20 0.38
HRH3 Q9Y5N1 1/20 0.38
KDM1A O60341 2/20 0.38
CNR1 P21554 2/20 0.38
GRM2 Q14416 1/20 0.38
AR P10275 1/20 0.37
NSD2 O96028 1/20 0.37
SCN10A Q9Y5Y9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8310064 0.99 BRS3 (0.49) BRS3GCGRMAPK14CYP11B1CYP11B2
SCHEMBL8110596 0.89 BRS3 (0.52) BRS3HRH3CNR1NSD2
SCHEMBL7919373 0.86 BRS3 (0.56) BRS3CYP11B1CYP11B2HRH3NSD2
Bromide SCHEMBL8310757 0.85 BRS3 (0.55) BRS3CYP11B1CYP11B2HRH3NSD2
SCHEMBL7927590 0.84 BRS3 (0.61) BRS3HRH3
SCHEMBL8107149 0.83 BRS3 (0.52) BRS3HRH3AR
Hydrochloric Acid SCHEMBL8307923 0.82 BRS3 (0.51) BRS3HRH3AR
SCHEMBL8112542 0.81 BRS3 (0.57) BRS3HRH3AR
SCHEMBL8105207 0.81 BRS3 (0.53) BRS3CYP11B1CYP11B2HRH3CNR1
SCHEMBL8097346 0.80 BRS3 (0.61) BRS3CYP11B1CYP11B2HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0986302-A1 A METHOD OF TREATING CANCER Merck & Co., Inc. (US) 2000-03-22 EP claimed
EP-0891333-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 1999-01-20 EP claimed
WO-1998054966-A1 A METHOD OF TREATING CANCER MERCK & CO., INC. (US) 1998-12-10 WO claimed
WO-1997036875-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 1997-10-09 WO claimed
EP-0986302-A1 A METHOD OF TREATING CANCER Merck & Co., Inc. (US) 2000-03-22 EP disclosed
WO-1998054966-A1 A METHOD OF TREATING CANCER MERCK & CO., INC. (US) 1998-12-10 WO disclosed