SCHEMBL8097549

SCHEMBL8097549

C[C@H](C(=O)c1ccc(F)cc1F)n1ncn(-c2ccc(OCC(F)(F)C(F)F)cc2)c1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 1/20 0.37
CYP17A1 P05093 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP19A1 P11511 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP11B1 P15538 1/20 0.37
CYP11B2 P19099 1/20 0.37
PTGS2 P35354 1/20 0.37
ABCG2 Q9UNQ0 1/20 0.37
CYP8B1 Q9UNU6 1/20 0.37
PPARD Q03181 10/20 0.36
PPARA Q07869 10/20 0.36
MAPT P10636 2/20 0.36
KDM4E B2RXH2 2/20 0.36
TSHR P16473 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
HTT P42858 3/20 0.35
SMN1; SMN2 Q16637 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8111202 0.85 KDM4E (0.37) CYP3A4CYP11B1CYP11B2KDM4ETSHR
SCHEMBL8097528 0.83 MAPT (0.41) PPARDPPARAMAPTKDM4EHTT
SCHEMBL8097580 0.82 MAPT (0.41) PPARDPPARAMAPTKDM4EHTT
SCHEMBL8097530 0.80 CYP3A4 (0.38) ABCB11CYP17A1CYP3A4CYP19A1CYP2C9
SCHEMBL8097526 0.80 CYP3A4 (0.38) ABCB11CYP17A1CYP3A4CYP19A1CYP2C9
SCHEMBL8106768 0.80 CYP3A4 (0.37) ABCB11CYP17A1CYP3A4CYP19A1CYP2C9
SCHEMBL8106771 0.80 CYP3A4 (0.37) ABCB11CYP17A1CYP3A4CYP19A1CYP2C9
SCHEMBL8718644 0.78 CYP3A4 (0.43) ABCB11CYP17A1CYP3A4CYP19A1CYP2C9
SCHEMBL8718648 0.78 CYP3A4 (0.43) ABCB11CYP17A1CYP3A4CYP19A1CYP2C9
SCHEMBL8111174 0.77 CYP3A4 (0.35) ABCB11CYP17A1CYP3A4CYP19A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1033367-A2 Process for the preparation of optically active triazole derivatives and their imidazolidin-2-one intermediates TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-09-06 EP disclosed
US-5677464-A Production of optically active triazole compounds and their intermediates TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-10-14 US disclosed
EP-0687672-A2 Production of optically active triazole compounds and their intermediates TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-12-20 EP disclosed