SCHEMBL8097556

SCHEMBL8097556

CNC(=O)Nc1ccc(-c2nc(N)cc(C3(S(C)(=O)=O)CCC3)n2)cc1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 6/20 0.42
MTOR P42345 5/20 0.42
PIK3CG P48736 1/20 0.42
PIP4K2A P48426 1/20 0.42
PIP4K2B P78356 1/20 0.42
PIK3CD O00329 8/20 0.40
KMT2A Q03164 1/20 0.39
AKT1 P31749 2/20 0.38
AKT2 P31751 2/20 0.38
ATR Q13535 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8098293 0.98 PIK3CA (0.42) PIK3CAMTORPIK3CGPIP4K2APIP4K2B
SCHEMBL8097448 0.96 PIK3CA (0.43) PIK3CAMTORPIK3CGPIP4K2APIP4K2B
SCHEMBL8092043 0.91 MTOR (0.49) PIK3CAMTORPIK3CGPIK3CDATR
SCHEMBL8090739 0.91 PIK3CA (0.40) PIK3CAMTORPIK3CGPIP4K2APIP4K2B
SCHEMBL8097252 0.90 CA12 (0.43) PIK3CAMTORPIK3CDKMT2AATR
SCHEMBL8093280 0.90 PIK3CA (0.41) PIK3CAMTORPIK3CGPIP4K2APIP4K2B
SCHEMBL8103635 0.89 ATR (0.39) PIK3CAMTORPIK3CDKMT2AAKT1
SCHEMBL8093447 0.88 MTOR (0.43) PIK3CAMTORPIK3CGPIP4K2APIP4K2B
SCHEMBL8098306 0.88 CA12 (0.42) PIK3CAMTORPIK3CD
SCHEMBL8091781 0.88 CA12 (0.43) PIK3CAMTORPIK3CDKMT2AATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed