SCHEMBL8103635

SCHEMBL8103635

CS(=O)(=O)C1(c2cc(N)nc(-c3ccc(NC(N)=O)cc3)n2)CCC1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ATR Q13535 3/20 0.39
KIF11 P52732 4/20 0.37
PIK3CD O00329 7/20 0.37
MEN1 O00255 3/20 0.37
ALDH1A1 P00352 3/20 0.37
MAPT P10636 3/20 0.37
HPGD P15428 3/20 0.37
KMT2A Q03164 3/20 0.37
KDM4E B2RXH2 2/20 0.37
RXFP1 Q9HBX9 2/20 0.37
MTOR P42345 1/20 0.36
PIK3CA P42336 2/20 0.35
AKT1 P31749 2/20 0.35
AKT2 P31751 2/20 0.35
NPSR1 Q6W5P4 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8083011 0.98 ATR (0.39) ATRKIF11PIK3CDMEN1ALDH1A1
SCHEMBL8083616 0.96 ATR (0.42) ATRKIF11PIK3CDMEN1ALDH1A1
SCHEMBL8097556 0.89 PIK3CA (0.42) ATRPIK3CDKMT2AMTORPIK3CA
SCHEMBL8097252 0.88 CA12 (0.43) ATRPIK3CDMEN1ALDH1A1MAPT
SCHEMBL8098293 0.87 PIK3CA (0.42) ATRPIK3CDMEN1ALDH1A1MAPT
SCHEMBL8098306 0.86 CA12 (0.42) PIK3CDALDH1A1MTORPIK3CACYP2C19
SCHEMBL8084829 0.86 ATR (0.41) ATRKIF11PIK3CDMEN1ALDH1A1
SCHEMBL8091781 0.85 CA12 (0.43) ATRPIK3CDMEN1ALDH1A1MAPT
SCHEMBL8099109 0.85 CA12 (0.43) PIK3CDMEN1ALDH1A1KMT2ACYP2C19
SCHEMBL8088889 0.85 PIK3CD (0.44) PIK3CDMEN1KMT2AMTORPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed