SCHEMBL8099469

SCHEMBL8099469

NS(=O)(=O)c1ccc(NS(=O)(=O)C(F)(F)F)c(Sc2ccc(Cl)cc2Cl)c1

nearest known ligand 0.63

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CA2 P00918 17/20 0.63
CA1 P00915 12/20 0.54
PTGS1 P23219 2/20 0.42
PTGS2 P35354 2/20 0.42
CA9 Q16790 1/20 0.41
CCR2 P41597 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8481841 1.00 CA2 (0.63) CA2CA1PTGS1PTGS2CA9
SCHEMBL8481837 0.99 CA2 (0.62) CA2CA1PTGS1PTGS2CA9
SCHEMBL8107827 0.89 CA2 (0.48) CA2CA1PTGS1PTGS2CA9
SCHEMBL7063507 0.85 CA2 (0.44) CA2CA1PTGS1PTGS2CA9
SCHEMBL4575696 0.84 PTGS1 (0.56) CA2CA1PTGS1PTGS2CA9
SCHEMBL8098906 0.82 PTGS1 (0.43) CA2CA1PTGS1PTGS2CA9
SCHEMBL8101068 0.81 PTGS1 (0.43) CA2CA1PTGS1PTGS2CA9
SCHEMBL7067324 0.81 CA2 (0.41) CA2CA1PTGS1PTGS2CA9
SCHEMBL8100682 0.81 PTGES2 (0.42) CA2CA1PTGS1PTGS2CA9
SCHEMBL8107826 0.80 CA2 (0.42) CA2CA1PTGS1PTGS2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0848703-B1 DERIVATIVES OF BENZOSULPHONAMIDES AS INHIBITORS OF THE ENZYME CYCLO-OXYGENASE II NYCOMED AUSTRIA GMBH (AT) 2000-09-27 EP disclosed
US-6004948-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS; SIDE EFFECT REDUCTION NYCOMED AUSTRIA GMBH (AT) 1999-12-21 US disclosed