SCHEMBL8099595

SCHEMBL8099595

COc1ccc(CCCNCCCc2ccccc2)cc1

nearest known ligand 0.68

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 0.68
MEN1 O00255 2/20 0.62
KMT2A Q03164 2/20 0.62
DRD2 P14416 3/20 0.62
DRD4 P21917 3/20 0.62
DRD3 P35462 3/20 0.62
ATM Q13315 1/20 0.59
CHRM2 P08172 1/20 0.59
ALDH1A1 P00352 1/20 0.58
LMNA P02545 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
LTA4H P09960 1/20 0.58
TDP1 Q9NUW8 1/20 0.58
L3MBTL1 Q9Y468 1/20 0.58
BCHE P06276 1/20 0.58
HTR2A P28223 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3621768 0.97 SIGMAR1 (0.70) SIGMAR1MEN1KMT2ADRD2DRD4
SCHEMBL6552032 0.92 MEN1 (0.71) SIGMAR1MEN1KMT2AATMCHRM2
SCHEMBL9520509 0.92 MEN1 (0.71) SIGMAR1MEN1KMT2AATMCHRM2
SCHEMBL9372179 0.90 SIGMAR1 (0.72) SIGMAR1MEN1KMT2AATMCHRM2
SCHEMBL4614753 0.89 MEN1 (0.71) MEN1KMT2AATMALDH1A1SMN1; SMN2
SCHEMBL5632470 0.87 LTA4H (0.69) SIGMAR1ALDH1A1LTA4HTDP1L3MBTL1
SCHEMBL275640 0.86 CHRM2 (0.59) SIGMAR1MEN1KMT2ACHRM2ALDH1A1
SCHEMBL5966301 0.85 TDP1 (0.75) SIGMAR1ALDH1A1LTA4HTDP1L3MBTL1
SCHEMBL12040566 0.85 TDP1 (0.75) SIGMAR1ALDH1A1LTA4HTDP1L3MBTL1
SCHEMBL6835324 0.84 CHRM2 (0.56) SIGMAR1CHRM2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057371-A TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS, GASTROINTESTINAL DISORDERS, DRUG ABUSE, ANGINA, MIGRAINE, HYPERTENSION AND DEPRESSION VIRGINIA COMMONWEALTH UNIVERSITY (US) 2000-05-02 US disclosed
EP-0591426-A1 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1994-04-13 EP disclosed
WO-1993000313-A2 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1993-01-07 WO disclosed
WO-1991009594-A1 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1991-07-11 WO disclosed