SCHEMBL8099744

SCHEMBL8099744

Nc1cc(C2(S(=O)(=O)c3ccncc3)CC2)nc(-c2ccc(NC(=O)NCCCO)cc2)n1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 10/20 0.40
PIK3CD O00329 5/20 0.37
PIK3CA P42336 3/20 0.37
MTOR P42345 2/20 0.37
ROCK2 O75116 2/20 0.36
ROCK1 Q13464 2/20 0.36
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.36
GLA P06280 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
PIK3CB P42338 1/20 0.35
PIK3CG P48736 1/20 0.35
PDGFRB P09619 1/20 0.35
KDR P35968 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8090241 0.95 NAMPT (0.43) NAMPTPIK3CDPIK3CAMTORROCK2
SCHEMBL8083986 0.92 CA2 (0.39) NAMPTPIK3CDPIK3CAMTORKDM4E
SCHEMBL8090391 0.91 CA1 (0.41) NAMPTPIK3CDPIK3CAMTOR
SCHEMBL8092289 0.91 CA1 (0.41) NAMPTPIK3CDPIK3CAMTORKDM4E
SCHEMBL8083655 0.90 NAMPT (0.43) NAMPTPIK3CDPIK3CAKDR
SCHEMBL8091160 0.89 NAMPT (0.38) NAMPTPIK3CDPIK3CAMTORKDM4E
SCHEMBL8104820 0.89 CA2 (0.38) NAMPTPIK3CDPIK3CAMTORKDM4E
SCHEMBL8083993 0.89 CA2 (0.38) NAMPTPIK3CDPIK3CAMTORKDM4E
SCHEMBL8084990 0.87 CA1 (0.40) NAMPTPIK3CDPIK3CAMTOR
SCHEMBL8091068 0.87 PIK3CD (0.42) PIK3CDPIK3CAMTORKDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed