SCHEMBL8090241

SCHEMBL8090241

Nc1cc(C2(S(=O)(=O)c3ccncc3)CC2)nc(-c2ccc(NC(=O)NCCO)cc2)n1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 9/20 0.43
PIK3CA P42336 6/20 0.41
MTOR P42345 3/20 0.41
PIK3CD O00329 7/20 0.39
PIK3CB P42338 1/20 0.39
PIK3CG P48736 1/20 0.39
ROCK2 O75116 2/20 0.37
ROCK1 Q13464 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8099744 0.95 NAMPT (0.40) NAMPTPIK3CAMTORPIK3CDPIK3CB
SCHEMBL8083655 0.92 NAMPT (0.43) NAMPTPIK3CAPIK3CD
SCHEMBL8098775 0.90 CA1 (0.43) NAMPTPIK3CAMTORPIK3CDPIK3CB
SCHEMBL8092406 0.89 PIK3CA (0.41) NAMPTPIK3CAMTORPIK3CDPIK3CB
SCHEMBL8084013 0.89 PIK3CA (0.41) NAMPTPIK3CAMTORPIK3CDPIK3CB
SCHEMBL8082005 0.89 PIK3CA (0.41) NAMPTPIK3CAMTORPIK3CDPIK3CB
SCHEMBL8099812 0.88 NAMPT (0.44) NAMPTPIK3CAPIK3CDROCK2ROCK1
SCHEMBL8099749 0.87 MTOR (0.40) NAMPTPIK3CAMTORPIK3CDPIK3CG
SCHEMBL8093138 0.87 NAMPT (0.40) NAMPTPIK3CAMTORPIK3CDPIK3CB
SCHEMBL8100146 0.87 CA1 (0.41) NAMPTPIK3CAMTORPIK3CDPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed