SCHEMBL8101092

SCHEMBL8101092

Cc1ccc(Oc2ccccc2N)c(C)c1

nearest known ligand 0.69

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.59
GAA P10253 2/20 0.59
SLC6A4 P31645 3/20 0.53
HTR1A P08908 2/20 0.50
HTR3A P46098 2/20 0.50
CYP3A4 P08684 1/20 0.46
TDP1 Q9NUW8 2/20 0.45
ADRA2B P18089 1/20 0.45
PTGS1 P23219 1/20 0.45
RCE1 Q9Y256 1/20 0.44
SLC6A2 P23975 2/20 0.44
SLC6A3 Q01959 2/20 0.44
KDM4E B2RXH2 1/20 0.44
MAPT P10636 1/20 0.44
CRHBP P24387 1/20 0.44
CRHR2 Q13324 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8737305 0.84 HTR1A (0.55) GAASLC6A4HTR1AHTR3ASLC6A2
SCHEMBL5607173 0.82 ALDH1A1 (0.56) ALDH1A1GAASLC6A4CYP3A4TDP1
SCHEMBL395415 0.82 ALDH1A1 (0.54) ALDH1A1GAASLC6A4CYP3A4TDP1
SCHEMBL29597724 0.82 ALDH1A1 (0.54) ALDH1A1GAASLC6A4CYP3A4TDP1
SCHEMBL31666386 0.82 HTR1A (0.50) ALDH1A1GAAHTR1AHTR3ACYP3A4
SCHEMBL4950654 0.82 HTR1A (0.50) ALDH1A1GAAHTR1AHTR3ACYP3A4
SCHEMBL9292115 0.81 ALDH1A1 (0.47) ALDH1A1GAASLC6A4TDP1ADRA2B
SCHEMBL8659962 0.81 IDO1 (0.53) ALDH1A1GAASLC6A4HTR1AHTR3A
Hydrochloric Acid SCHEMBL10423028 0.80 ALDH1A1 (0.45) ALDH1A1GAASLC6A4HTR1AHTR3A
Hydrochloric Acid SCHEMBL10423771 0.79 ALDH1A1 (0.52) ALDH1A1GAASLC6A4HTR1AHTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0848703-B1 DERIVATIVES OF BENZOSULPHONAMIDES AS INHIBITORS OF THE ENZYME CYCLO-OXYGENASE II NYCOMED AUSTRIA GMBH (AT) 2000-09-27 EP disclosed
US-6004948-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS; SIDE EFFECT REDUCTION NYCOMED AUSTRIA GMBH (AT) 1999-12-21 US disclosed
EP-0848703-A1 DERIVATIVES OF BENZOSULPHONAMIDES AS INHIBITORS OF THE ENZYME CYCLO-OXYGENASE II Nycomed Austria GmbH (AT) 1998-06-24 EP disclosed
WO-1997003953-A1 DERIVATIVES OF BENZOSULPHONAMIDES AS INHIBITORS OF THE ENZYME CYCLO-OXYGENASE II NYCOMED AUSTRIA GMBH (AT) 1997-02-06 WO disclosed