SCHEMBL8101162

SCHEMBL8101162

CCNCCNC(=O)c1ccc(NC(C)=O)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.65
NFKB1 P19838 1/20 0.65
KCNH2 Q12809 1/20 0.65
SMN1; SMN2 Q16637 4/20 0.63
POLB P06746 3/20 0.63
CYP3A4 P08684 1/20 0.63
THRB P10828 1/20 0.63
BLM P54132 1/20 0.63
ATM Q13315 1/20 0.63
HTT P42858 3/20 0.58
TP53 P04637 1/20 0.53
HIF1A Q16665 1/20 0.53
CACNA1B Q00975 1/20 0.53
APBA1 Q02410 1/20 0.53
EPHX2 P34913 1/20 0.52
NR1H4 Q96RI1 1/20 0.52
NAMPT P43490 1/20 0.51
HDAC3 O15379 1/20 0.48
HDAC4 P56524 1/20 0.48
HDAC1 Q13547 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5508324 0.85 ALDH1A1 (0.70) ALDH1A1NFKB1KCNH2SMN1; SMN2POLB
SCHEMBL12368426 0.85 ALDH1A1 (0.65) ALDH1A1NFKB1KCNH2SMN1; SMN2POLB
SCHEMBL19013029 0.84 MEN1 (0.63) ALDH1A1SMN1; SMN2THRBHTTTP53
SCHEMBL5502874 0.83 SMN1; SMN2 (0.79) ALDH1A1NFKB1KCNH2SMN1; SMN2POLB
SCHEMBL22458558 0.82 SMN1; SMN2 (0.60) ALDH1A1NFKB1KCNH2SMN1; SMN2POLB
SCHEMBL5506823 0.81 SMN1; SMN2 (0.77) ALDH1A1NFKB1KCNH2SMN1; SMN2POLB
SCHEMBL10755434 0.81 SMN1; SMN2 (0.63) ALDH1A1NFKB1KCNH2SMN1; SMN2POLB
SCHEMBL11196763 0.81 ALDH1A1 (0.64) ALDH1A1NFKB1KCNH2SMN1; SMN2POLB
SCHEMBL13015281 0.80 CD274 (0.56) ALDH1A1NFKB1KCNH2SMN1; SMN2POLB
SCHEMBL10872851 0.80 LMNA (0.69) ALDH1A1SMN1; SMN2POLBCYP3A4HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0734526-A4 MALEIMIDE ADDUCT CONJUGATES OF PROCAINAMIDE AND NAPA ROCHE DIAGNOSTICS CORP (US) 2000-03-29 EP disclosed
EP-0734526-A1 MALEIMIDE ADDUCT CONJUGATES OF PROCAINAMIDE AND NAPA BOEHRINGER MANNHEIM CORPORATION (US) 1996-10-02 EP disclosed
US-5439798-A Immunoassay; competitive binding; quantitative analysis BOEHRINGER MANNHEIM CORPORATION (US) 1995-08-08 US disclosed
WO-1995016894-A1 MALEIMIDE ADDUCT CONJUGATES OF PROCAINAMIDE AND NAPA BOEHRINGER MANNHEIM CORPORATION (US) 1995-06-22 WO disclosed