Morpholine

Morpholine

SCHEMBL8101591

C1COCCN1.CC(C)NC(=O)CN1CCNCC1.CC(O)N1CCNCC1.O=C(CN1CCNCC1)N1CCCC1

nearest known ligand 0.59

Full drug profile on Sugi Atlas →

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 2/20 0.59
CHRM3 P20309 2/20 0.59
ALDH1A1 P00352 4/20 0.44
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39
HSD17B10 Q99714 1/20 0.39
BIRC2 Q13490 1/20 0.38
SIGMAR1 Q99720 3/20 0.36
GAA P10253 2/20 0.35
KDM4E B2RXH2 4/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
PKM P14618 1/20 0.34
NPC1 O15118 1/20 0.34
TDP1 Q9NUW8 1/20 0.33
POLB P06746 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C19 P33261 1/20 0.33
LMNA P02545 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8729488 0.86 CHRM5 (0.79) CHRM5CHRM3ALDH1A1BIRC2SIGMAR1
SCHEMBL255190 0.77 CHRM5 (1.00) CHRM5CHRM3ALDH1A1SIGMAR1GAA
SCHEMBL6963350 0.72 GAA (0.63) CHRM5CHRM3ALDH1A1ALOX15TSHR
Morpholine SCHEMBL8725832 0.72 MEN1 (0.44) CHRM5CHRM3GAAKDM4ESMN1; SMN2
SCHEMBL209616 0.72 GAA (0.63) CHRM5CHRM3ALDH1A1ALOX15TSHR
SCHEMBL255444 0.71 HSD17B10 (0.69) ALDH1A1ALOX15TSHRHSD17B10GAA
SCHEMBL2073211 0.71 HSD17B10 (0.69) ALDH1A1ALOX15TSHRHSD17B10GAA
SCHEMBL7720951 0.71 CHRM5 (0.64) CHRM5CHRM3ALDH1A1ALOX15TSHR
SCHEMBL254801 0.71 GAA (0.67) CHRM5CHRM3ALDH1A1ALOX15TSHR
Hydrochloric Acid SCHEMBL27822626 0.71 GAA (0.61) CHRM5CHRM3ALDH1A1ALOX15TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973936-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC AMINOTHIOETHER ACIDS ELI LILLY AND COMPANY (US) 2000-01-26 EP disclosed
WO-1998046786-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC AMINOTHIOETHER ACIDS ELI LILLY AND COMPANY (US) 1998-10-22 WO disclosed