SCHEMBL8101972

SCHEMBL8101972

COc1cccc([C@@H]2C[C@H]2C(=O)N(C)OC)c1

nearest known ligand 0.60

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 2/20 0.60
GPR88 Q9GZN0 2/20 0.49
HTR2A P28223 2/20 0.48
HTR2C P28335 2/20 0.48
HTR2B P41595 2/20 0.48
EPHX2 P34913 1/20 0.46
APP P05067 1/20 0.44
CHRM2 P08172 1/20 0.43
CHRM1 P11229 1/20 0.43
CHRM3 P20309 1/20 0.43
TRPM5 Q9NZQ8 1/20 0.43
DGAT2 Q96PD7 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MCL1 Q07820 2/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
GLA P06280 1/20 0.41
GAA P10253 1/20 0.41
HPGD P15428 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6320354 1.00 SLC9A1 (0.60) SLC9A1GPR88HTR2AHTR2CHTR2B
SCHEMBL9382461 0.85 SLC9A1 (0.45) SLC9A1GPR88EPHX2APPMCL1
SCHEMBL1223675 0.84 SLC9A1 (0.53) SLC9A1GPR88HTR2AHTR2CHTR2B
SCHEMBL1223671 0.84 SLC9A1 (0.53) SLC9A1GPR88HTR2AHTR2CHTR2B
SCHEMBL5675828 0.84 GPR88 (0.46) SLC9A1GPR88HTR2AHTR2CHTR2B
SCHEMBL6250729 0.83 MAPT (0.51) GPR88EPHX2L3MBTL1MCL1ALDH1A1
SCHEMBL17590033 0.83 MCL1 (0.55) SLC9A1GPR88EPHX2APPTRPM5
SCHEMBL15208924 0.83 MCL1 (0.55) SLC9A1GPR88EPHX2APPTRPM5
SCHEMBL17146213 0.83 MCL1 (0.55) SLC9A1GPR88EPHX2APPTRPM5
SCHEMBL13929891 0.83 MCL1 (0.55) SLC9A1GPR88EPHX2APPTRPM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0747346-B1 N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL MYERS SQUIBB CO (US) 2000-02-16 EP disclosed
US-5889031-A CONTROLLING CIRCADIAN RHYTHMS BRISTOL-MYERS SQUIBB COMPNAY (US) 1999-03-30 US disclosed
US-5753709-A N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL-MYERS SQUIBB COMPANY (US) 1998-05-19 US disclosed
EP-0747346-A2 N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL-MYERS SQUIBB COMPANY (US) 1996-12-11 EP disclosed