SCHEMBL8102406

SCHEMBL8102406

COC(=O)N1CC2CC1CN(Cc1ccccc1)C2

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.58
S1PR5 Q9H228 2/20 0.44
S1PR1 P21453 1/20 0.44
PSEN1 P49768 1/20 0.43
PSEN2 P49810 1/20 0.43
APH1B Q8WW43 1/20 0.43
NCSTN Q92542 1/20 0.43
APH1A Q96BI3 1/20 0.43
PSENEN Q9NZ42 1/20 0.43
ALDH1A1 P00352 2/20 0.43
CYP2D6 P10635 1/20 0.43
FUCA1 P04066 2/20 0.42
BCHE P06276 2/20 0.41
ACHE P22303 1/20 0.41
MAOB P27338 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL927653 0.86 HSD11B1 (0.55) HSD11B1S1PR5S1PR1FUCA1ACHE
SCHEMBL4318880 0.85 HSD11B1 (0.65) HSD11B1S1PR5S1PR1ALDH1A1FUCA1
SCHEMBL928056 0.80 HSD11B1 (0.58) HSD11B1S1PR5S1PR1ALDH1A1FUCA1
SCHEMBL2959552 0.78 HSD11B1 (0.46) HSD11B1S1PR5S1PR1ALDH1A1
SCHEMBL3237901 0.76 HSD11B1 (0.44) HSD11B1S1PR5S1PR1ACHEKMT2A
SCHEMBL6335547 0.75 HSD11B1 (0.51) HSD11B1S1PR5S1PR1FUCA1ACHE
SCHEMBL9055722 0.75 S1PR5 (0.50) S1PR5S1PR1ALDH1A1CYP2D6FUCA1
SCHEMBL20587395 0.75 AGTR2 (0.48) HSD11B1S1PR5S1PR1PSEN1PSEN2
SCHEMBL10480299 0.75 HSD11B1 (0.49) HSD11B1S1PR5S1PR1FUCA1ACHE
SCHEMBL6749184 0.75 S1PR5 (0.50) HSD11B1S1PR5S1PR1ALDH1A1FUCA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153608-A Isoquinoline derivatives and drugs NIPPON SHINYAKU CO., LTD. (JP) 2000-11-28 US disclosed
EP-0885888-A1 ISOQUINOLINE DERIVATIVES AND DRUGS NIPPON SHINYAKU COMPANY, LIMITED (JP) 1998-12-23 EP disclosed