SCHEMBL8102643

SCHEMBL8102643

C=CCOC(=O)CSC1CC(=O)N1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.37
ALDH1A1 P00352 4/20 0.36
GAA P10253 2/20 0.36
NPSR1 Q6W5P4 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.33
CYP3A4 P08684 1/20 0.33
CA1 P00915 3/20 0.32
CA2 P00918 3/20 0.32
EPHX2 P34913 1/20 0.32
PKM P14618 1/20 0.32
TDP1 Q9NUW8 2/20 0.32
HSD17B10 Q99714 1/20 0.32
ITGB3 P05106 1/20 0.32
ITGB2 P05107 1/20 0.32
ITGB1 P05556 1/20 0.32
ITGAV P06756 1/20 0.32
ITGA2B P08514 1/20 0.32
ITGA5 P08648 1/20 0.32
ITGB5 P18084 1/20 0.32
ITGAL P20701 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8104182 0.84 TSHR (0.44) TSHRALDH1A1GAANPSR1SMN1; SMN2
SCHEMBL8441196 0.79 NPSR1 (0.35) TSHRNPSR1SMN1; SMN2CYP3A4CA1
SCHEMBL8300761 0.73 SNCA (0.42) TSHRALDH1A1CYP3A4CA1CA2
SCHEMBL7716010 0.71
Allyl Alcohol SCHEMBL8437400 0.71 SNCA (0.40) TSHRALDH1A1CYP3A4CA1CA2
SCHEMBL31122206 0.68 TSHR (0.47) TSHRALDH1A1GAANPSR1SMN1; SMN2
SCHEMBL10715577 0.65
SCHEMBL10842299 0.64
SCHEMBL7578576 0.64 TSHR (0.43) TSHRALDH1A1GAANPSR1SMN1; SMN2
SCHEMBL6328278 0.62 ALDH1A1 (0.36) TSHRALDH1A1GAASMN1; SMN2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6071899-A Azetidinone derivatives for the treatment of atherosclerosis SMITHKLINE BEECHAM P.L.C. (GB) 2000-06-06 US disclosed
EP-0788478-A1 AZETIDINONE DERIVATIVES FOR THE TREATMENT OF ATHEROSCLEROSIS SMITHKLINE BEECHAM PLC (GB) 1997-08-13 EP disclosed
WO-1996013484-A1 AZETIDINONE DERIVATIVES FOR THE TREATMENT OF ATHEROSCLEROSIS SMITHKLINE BEECHAM PLC (GB) 1996-05-09 WO disclosed