SCHEMBL8102656

SCHEMBL8102656

ClCCN1CCN(c2ccc(Cl)cc2)CC1

nearest known ligand 0.63

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.63
GAA P10253 2/20 0.63
SIGMAR1 Q99720 3/20 0.59
DRD4 P21917 3/20 0.59
HTR1A P08908 7/20 0.56
DRD2 P14416 6/20 0.56
HTR2A P28223 4/20 0.56
DRD3 P35462 4/20 0.56
TMEM97 Q5BJF2 2/20 0.56
MAPT P10636 2/20 0.56
DRD1 P21728 3/20 0.55
DRD5 P21918 3/20 0.55
SLC6A2 P23975 2/20 0.55
SLC6A4 P31645 2/20 0.55
ALDH1A1 P00352 1/20 0.54
HTR7 P34969 1/20 0.54
CACNA1G O43497 1/20 0.52
SLC6A3 Q01959 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5179759 0.89 KDM4E (0.69) KDM4EGAASIGMAR1DRD4HTR1A
Hydrochloric Acid SCHEMBL11622828 0.87 KDM4E (0.67) KDM4EGAASIGMAR1DRD4HTR1A
SCHEMBL18754269 0.86 KDM4E (0.75) KDM4EGAASIGMAR1DRD4HTR1A
SCHEMBL13079491 0.85 KDM4E (0.78) KDM4EGAASIGMAR1DRD4HTR1A
SCHEMBL2093634 0.83 KDM4E (0.61) KDM4EGAASIGMAR1DRD4HTR1A
SCHEMBL7739933 0.83 MAPT (0.61) KDM4EGAASIGMAR1DRD4HTR1A
SCHEMBL4400393 0.83 KDM4E (0.61) KDM4EGAASIGMAR1DRD4HTR1A
SCHEMBL6184036 0.83 MAPT (0.58) GAASIGMAR1DRD4HTR1ADRD2
SCHEMBL10366646 0.83 KDM4E (0.61) KDM4EGAASIGMAR1DRD4HTR1A
SCHEMBL5836202 0.82 KCNH2 (0.69) KDM4ESIGMAR1DRD4HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0810206-B1 Substituted 2-naphthoylguanidines, process for their preparation, their use as medicament or diagnostic agent and medicament containing them HOECHST AG (DE) 2000-12-27 EP disclosed
US-6087304-A ANTIARRHYTHMIC PHARMACEUTICALS HAVING A CARDIOPROTECTIVE COMPONENT FOR INFARCT PROPHYLAXIS AND INFARCT TREATMENT AND FOR THE TREATMENT OF ANGINA PECTORIS HOECHST AKTIENGESELLSCHAFT (DE) 2000-07-11 US disclosed
EP-0810206-A1 Substituted 2-naphtoylguanidines, process for their preparation, their use as medicament or diagnostic agent and medicament containing them HOECHST AKTIENGESELLSCHAFT (DE) 1997-12-03 EP disclosed