SCHEMBL8102926

SCHEMBL8102926

COc1ncc(F)c2nnc(SCc3ccccc3)n12

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.43
RAB9A P51151 5/20 0.43
NPC1 O15118 4/20 0.43
TSHR P16473 1/20 0.43
LMNA P02545 2/20 0.42
KDM4E B2RXH2 2/20 0.40
SIRT2 Q8IXJ6 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
GPBAR1 Q8TDU6 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8103143 0.75 ALDH1A1 (0.49) ALDH1A1RAB9ANPC1TSHRLMNA
SCHEMBL9536661 0.68 ALDH1A1 (0.44) ALDH1A1RAB9ANPC1TSHRLMNA
SCHEMBL8111879 0.67 MAPT (0.43) ALDH1A1RAB9ANPC1TSHRLMNA
SCHEMBL17668058 0.64 PKM (0.46) ALDH1A1RAB9ANPC1TSHRLMNA
SCHEMBL9642664 0.63 ALDH1A1 (0.53) ALDH1A1RAB9ANPC1TSHRLMNA
SCHEMBL9642141 0.63 ALDH1A1 (0.50) ALDH1A1RAB9ANPC1TSHRLMNA
SCHEMBL4212033 0.63 ALDH1A1 (0.70) ALDH1A1RAB9ANPC1TSHRKDM4E
SCHEMBL9642193 0.63 ALDH1A1 (0.47) ALDH1A1RAB9ANPC1TSHRKDM4E
SCHEMBL8111887 0.63 ALDH1A1 (0.49) ALDH1A1RAB9ANPC1TSHRLMNA
SCHEMBL9640970 0.63 ALDH1A1 (0.49) ALDH1A1RAB9ANPC1TSHRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0678094-B1 2-ALKOXY-4-HYDRAZINOPYRIMIDINE COMPOUNDS AND THEIR USE IN THE PREPARATION OF 5-ALKOXY[1,2,4]TRIAZOLO[4,3-C]PYRIMIDINE-3(2H)-THIONE COMPOUNDS DOW AGROSCIENCES LLC (US) 2000-05-03 EP disclosed
EP-0678093-B1 5-ALKOXY-1,2,4-TRIAZOLO[4,3-C]PYRIMIDINE-3(2H)-THIONE COMPOUNDS AND THEIR USE IN THE PREPARATION OF 5-ALKOXY-1,2,4-TRIAZOLO[1,5-C]PYRIMIDINE-2(3H)-THIONE AND 3-HYDROCARBYLTHIO-5-ALKOXY-1,2,4-TRIAZOLO[4,3-C]PYRIMIDINE COMPOUNDS DOW AGROSCIENCES LLC (US) 2000-01-05 EP disclosed
US-5563269-A 2-alkoxy-4-hydrazinopyrimidine compounds and their use in the preparation of 5-alkoxy-1,2,4-triazolo(4,3-C)-pyrimidine-3 (2H)-thione compounds DOWELANCO (US) 1996-10-08 US disclosed
US-5480991-A 2-Alkoxy-4-hydroazinopyrimidine compounds and their use in the preparation of 5-alkoxy-1,2,4-triazolo[4,3-c]pyrimidine-3(2H)-thione compounds DOWELANCO (US) 1996-01-02 US disclosed
US-5461153-A 2-alkoxy-4-hydrazinopyrimidine compounds DOWELANCO (US) 1995-10-24 US disclosed