SCHEMBL8103130

SCHEMBL8103130

CC(=O)OCc1ccc(NC(=O)C(NC(=O)OC(C)(C)C)c2ccc3c(c2)C(C)(C)CCC3(C)C)cc1

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 4/20 0.42
CYP26A1 O43174 2/20 0.40
CYP26B1 Q9NR63 2/20 0.40
ALDH1A1 P00352 1/20 0.38
CYP3A4 P08684 1/20 0.38
TSHR P16473 1/20 0.38
JAK2 O60674 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8100687 0.88 CYP3A4 (0.47) BACE1ALDH1A1CYP3A4TSHRJAK2
SCHEMBL8100983 0.86 RARB (0.44) CYP26A1CYP26B1ALDH1A1CYP3A4TSHR
SCHEMBL8106743 0.86 MEN1 (0.42) CYP26A1CYP26B1ALDH1A1CYP3A4TSHR
SCHEMBL8757257 0.85 RARB (0.40) BACE1CYP26A1CYP26B1ALDH1A1CYP3A4
SCHEMBL8748829 0.84 RARB (0.55) CYP26A1CYP26B1ALDH1A1CYP3A4TSHR
SCHEMBL8102431 0.83 RARB (0.43) CYP26A1CYP26B1ALDH1A1CYP3A4TSHR
SCHEMBL8093042 0.82 RORC (0.45) CYP26A1CYP26B1ALDH1A1CYP3A4TSHR
SCHEMBL8093059 0.82 CYP26A1 (0.44) CYP26A1CYP26B1ALDH1A1CYP3A4TSHR
SCHEMBL8561391 0.81 CTSS (0.48) BACE1CYP3A4
SCHEMBL8093109 0.79 RARG (0.43) CYP26A1CYP26B1ALDH1A1CYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6051243-A USEFUL IN THE TOPICAL AND SYSTEMIC TREATMENT OF DERMATOLOGICAL CONDITIONS ASSOCIATED WITH A KERATINIZATION DISORDER, DERMATOLOGICAL CONDITIONS (AND THE LIKE) INCLUDING AN INFLAMMATORY AND/OR IMMUNOALLERGIC COMPONENT CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES (FR) 2000-04-18 US disclosed