SCHEMBL8103554

SCHEMBL8103554

COc1ccc(C(=O)CBr)cc1.O=C(CBr)c1ccc(-c2ccccc2)cc1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 3/20 0.77
PTPN1 P18031 2/20 0.74
KMT2A Q03164 2/20 0.60
CYP3A4 P08684 2/20 0.60
MEN1 O00255 1/20 0.60
NPC1 O15118 2/20 0.58
RAB9A P51151 2/20 0.58
ALDH1A1 P00352 2/20 0.55
POLB P06746 2/20 0.55
CTDSP1 Q9GZU7 2/20 0.55
MAPT P10636 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
L3MBTL1 Q9Y468 2/20 0.54
CES2 O00748 1/20 0.54
CES1 P23141 1/20 0.54
HSD11B1 P28845 1/20 0.54
LMNA P02545 1/20 0.54
HDAC3 O15379 1/20 0.53
HDAC4 P56524 1/20 0.53
HDAC1 Q13547 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7390281 0.93 GSK3B (0.89) GSK3BPTPN1NPC1RAB9AMAPT
SCHEMBL202055 0.88 GSK3B (1.00) GSK3BPTPN1NPC1RAB9AALDH1A1
SCHEMBL16203309 0.87 KMT2A (0.68) KMT2ACYP3A4MEN1NPC1RAB9A
Ammonia Solution, Strong SCHEMBL17626749 0.86 GSK3B (0.96) GSK3BPTPN1NPC1RAB9AALDH1A1
SCHEMBL316871 0.86 GSK3B (1.00) GSK3BPTPN1RAB9AALDH1A1MAPT
SCHEMBL22004470 0.86 GSK3B (1.00) GSK3BPTPN1RAB9AALDH1A1MAPT
SCHEMBL4328500 0.84 GSK3B (0.73) GSK3BPTPN1KMT2ANPC1RAB9A
SCHEMBL2773360 0.83 GSK3B (0.89) GSK3BPTPN1NPC1RAB9AALDH1A1
SCHEMBL1694670 0.83 NPC1 (0.63) KMT2ACYP3A4MEN1NPC1RAB9A
SCHEMBL31357491 0.83 MAPT (0.78) KMT2ACYP3A4MEN1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973936-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC AMINOTHIOETHER ACIDS ELI LILLY AND COMPANY (US) 2000-01-26 EP disclosed
WO-1998046786-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC AMINOTHIOETHER ACIDS ELI LILLY AND COMPANY (US) 1998-10-22 WO disclosed