SCHEMBL8103669

SCHEMBL8103669

CS(=O)(=O)c1cc(COC(=O)N=C(N)N)ccc1Oc1cccc2cccnc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44
CA14 Q9ULX7 1/20 0.44
KDM4E B2RXH2 4/20 0.43
MAPT P10636 3/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
TDP1 Q9NUW8 2/20 0.43
PRSS1 P07477 1/20 0.42
ACR P10323 1/20 0.42
ALDH1A1 P00352 1/20 0.41
AOC3 Q16853 7/20 0.41
LMNA P02545 2/20 0.40
MAPK1 P28482 1/20 0.40
HDAC6 Q9UBN7 1/20 0.39
POLB P06746 1/20 0.39
HSD17B10 Q99714 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7995604 0.83 AOC3 (0.40) ALDH1A1AOC3
Hydrochloric Acid SCHEMBL8007034 0.83 AOC3 (0.41) ALDH1A1AOC3
Hydrochloric Acid SCHEMBL8104379 0.83 AOC3 (0.41) ALDH1A1AOC3
Water SCHEMBL8095247 0.76 SCN9A (0.40) KDM4EMAPTALDH1A1LMNAMAPK1
SCHEMBL8832381 0.73 MAPT (0.48) CA12CA1CA2CA9CA14
SCHEMBL8005829 0.73 PPARG (0.37)
Hydrochloric Acid SCHEMBL8102087 0.72 PPARG (0.36) AOC3
SCHEMBL8007047 0.69 SLC9A1 (0.60) AOC3
SCHEMBL8004007 0.69 C5AR1 (0.37) CA2
SCHEMBL8180320 0.69 SLC9A1 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0748795-B1 Substituted benzyloxycarbonyl guanidines as Na+/H+ exchange inhibitors, process for their preparation, their use as medicinal or diagnostic agents as well as medicament containing them HOECHST AG (DE) 2000-08-23 EP disclosed
EP-0748795-A2 Substituted benzyloxycarbonyl guanidines as Na+/H+ exchange inhibitors, process for their preparation, their use as medicinal or diagnostic agents as well as medicament containing them HOECHST AKTIENGESELLSCHAFT (DE) 1996-12-18 EP disclosed