SCHEMBL8005829

SCHEMBL8005829

Cc1ccc2cc(Oc3ccc(COC(=O)N=C(N)N)cc3S(C)(=O)=O)ccc2n1

nearest known ligand 0.41

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.37
SCN9A Q15858 1/20 0.34
GCK P35557 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8102087 0.99 PPARG (0.36) PPARGSCN9AGCK
SCHEMBL7995604 0.86 AOC3 (0.40) PPARGSCN9A
Hydrochloric Acid SCHEMBL8104379 0.85 AOC3 (0.41) PPARGSCN9A
Hydrochloric Acid SCHEMBL8007034 0.85 AOC3 (0.41) PPARGSCN9A
SCHEMBL8006634 0.83 PPARG (0.38) PPARGSCN9A
Hydrochloric Acid SCHEMBL8611682 0.83 PPARG (0.38) PPARGSCN9A
Water SCHEMBL8095247 0.78 SCN9A (0.40) PPARGSCN9A
SCHEMBL8880848 0.74 PDE4B (0.43) SCN9AGCK
SCHEMBL8103669 0.73 CA12 (0.44)
SCHEMBL7995599 0.71 ALDH1A1 (0.41) PPARGSCN9AGCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6022899-A EFFECTIVE INHIBITORS OF THE CELLULAR SODIUM PROTON ANTIPORTER HOECHST AKTIENGESELLSCHAFT (DE) 2000-02-08 US disclosed
US-5753710-A INHIBITORS OF THE CELLULAR SODIUM PROTON ANTIPORTER HOECHST AKTIENGESELLSCHAFT (DE) 1998-05-19 US disclosed