SCHEMBL8103916

SCHEMBL8103916

Oc1ccc2[nH]cc(C3CCN(N4CCCCC4)CC3)c2c1

nearest known ligand 0.71

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.71
CYP3A4 P08684 1/20 0.71
CYP2D6 P10635 1/20 0.71
CYP2C9 P11712 1/20 0.71
THPO P40225 1/20 0.71
MAPT P10636 1/20 0.60
BLM P54132 1/20 0.60
NPSR1 Q6W5P4 1/20 0.60
HTR1D P28221 3/20 0.50
HTR1B P28222 3/20 0.50
OPRM1 P35372 1/20 0.49
OPRK1 P41145 1/20 0.49
OPRL1 P41146 1/20 0.49
ADRA1D P25100 3/20 0.47
HSD11B1 P28845 1/20 0.46
HTR1A P08908 1/20 0.46
HTR1F P30939 1/20 0.46
SLC6A4 P31645 2/20 0.46
APP P05067 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18622640 0.86 CYP1A2 (0.69) CYP1A2CYP3A4CYP2D6CYP2C9THPO
SCHEMBL8109749 0.84 OPRM1 (0.62) CYP1A2CYP3A4CYP2D6CYP2C9THPO
SCHEMBL8096608 0.84 HTR1D (0.53) CYP1A2CYP3A4CYP2D6CYP2C9THPO
SCHEMBL8109656 0.84 OPRM1 (0.68) HTR1BOPRM1OPRK1OPRL1ADRA1D
SCHEMBL3546728 0.83 CYP1A2 (1.00) CYP1A2CYP3A4CYP2D6CYP2C9THPO
SCHEMBL30908918 0.83 CYP1A2 (1.00) CYP1A2CYP3A4CYP2D6CYP2C9THPO
SCHEMBL8103895 0.81 SLC6A4 (0.69) HTR1BHTR1ASLC6A4
SCHEMBL5705057 0.79 CYP1A2 (0.72) CYP1A2CYP3A4CYP2D6CYP2C9THPO
SCHEMBL3549500 0.79 CYP1A2 (0.68) CYP1A2CYP3A4CYP2D6CYP2C9THPO
SCHEMBL8103912 0.78 CYP1A2 (0.54) CYP1A2CYP3A4CYP2D6CYP2C9THPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6143744-A Sulfamide-metalloprotease inhibitors SYNTEX (U.S.A.) INC. (US) 2000-11-07 US disclosed
US-6130220-A ENZYME INHIBITORS SYNTEX (USA) INC. (US) 2000-10-10 US disclosed
US-5998412-A ANTIARTHRITIC AGENTS; OSTEOPOROSIS SYNTEX (U.S.A.) INC. (US) 1999-12-07 US disclosed