SCHEMBL8104322

SCHEMBL8104322

O=C(NC[C@@H]1C[C@H]1c1cccc(Cl)c1)C1CC1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.54
HTR2C P28335 2/20 0.54
HTR2B P41595 2/20 0.54
CNR1 P21554 2/20 0.49
MTNR1A P48039 6/20 0.47
MTNR1B P49286 6/20 0.47
ALDH1A1 P00352 1/20 0.44
SLC9A1 P19634 1/20 0.43
DPP4 P27487 1/20 0.42
DPP8 Q6V1X1 1/20 0.42
DPP9 Q86TI2 1/20 0.42
DPP7 Q9UHL4 1/20 0.42
CHRM1 P11229 1/20 0.42
CHRM3 P20309 1/20 0.42
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8098094 0.84 HTR2C (0.54) HTR2AHTR2CHTR2BCNR1MTNR1A
SCHEMBL8098093 0.84 HTR2C (0.54) HTR2AHTR2CHTR2BCNR1MTNR1A
SCHEMBL8102597 0.84 HTR2C (0.56) HTR2AHTR2CHTR2BCNR1MTNR1A
SCHEMBL8102591 0.84 HTR2C (0.56) HTR2AHTR2CHTR2BCNR1MTNR1A
SCHEMBL8102766 0.81 HTR2A (0.56) HTR2AHTR2CHTR2BMTNR1AMTNR1B
SCHEMBL8096201 0.80 HTR2C (0.51) HTR2AHTR2CHTR2BCNR1MTNR1A
SCHEMBL8096202 0.80 HTR2C (0.51) HTR2AHTR2CHTR2BCNR1MTNR1A
SCHEMBL24737408 0.75 HTR2A (0.62) HTR2AHTR2CHTR2BSLC9A1
SCHEMBL30711641 0.74 HTR2C (0.70) HTR2AHTR2CHTR2BSLC9A1
SCHEMBL27033783 0.74 HTR2C (0.70) HTR2AHTR2CHTR2BSLC9A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0747346-B1 N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL MYERS SQUIBB CO (US) 2000-02-16 EP disclosed
EP-0747346-A2 N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL-MYERS SQUIBB COMPANY (US) 1996-12-11 EP disclosed