SCHEMBL8104823

SCHEMBL8104823

Nc1cc(C2(S(=O)(=O)c3ccccc3)CCC2)nc(-c2ccc(NC(=O)NCCF)cc2)n1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.39
CA12 O43570 2/20 0.39
CA1 P00915 2/20 0.39
CA4 P22748 2/20 0.39
CA7 P43166 2/20 0.39
CA9 Q16790 2/20 0.39
NAMPT P43490 5/20 0.38
PIK3CA P42336 6/20 0.38
MTOR P42345 6/20 0.38
PIK3CD O00329 4/20 0.37
CYP2C9 P11712 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MAPT P10636 1/20 0.36
HTT P42858 1/20 0.36
AKT1 P31749 1/20 0.35
AKT2 P31751 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8091717 0.96 CA2 (0.40) CA2CA12CA1CA4CA7
SCHEMBL8083998 0.92 CA2 (0.39) CA2CA12CA1CA4CA7
SCHEMBL8084013 0.92 PIK3CA (0.41) CA2CA12CA1CA4CA7
SCHEMBL8104820 0.91 CA2 (0.38) CA2CA12CA1CA4CA7
SCHEMBL8092406 0.90 PIK3CA (0.41) CA2CA12CA1CA4CA7
SCHEMBL8089052 0.90 CA2 (0.41) CA2CA12CA1CA4CA7
SCHEMBL8083993 0.89 CA2 (0.38) CA2CA12CA1CA4CA7
SCHEMBL8099632 0.88 CA1 (0.42) CA2CA12CA1CA4CA7
SCHEMBL8092385 0.88 PIK3CD (0.41) CA2CA12CA1CA4CA7
SCHEMBL8100085 0.87 NAMPT (0.38) CA2CA12CA1CA4CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed