SCHEMBL8099632

SCHEMBL8099632

Cc1ccc(S(=O)(=O)C2(c3cc(N)nc(-c4ccc(NC(=O)NCCF)cc4)n3)CC2)cc1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.42
CA2 P00918 3/20 0.42
CA12 O43570 2/20 0.42
CA4 P22748 2/20 0.42
CA7 P43166 2/20 0.42
CA9 Q16790 2/20 0.42
ALDH1A1 P00352 1/20 0.40
PIK3CD O00329 4/20 0.38
PIK3CA P42336 3/20 0.38
MTOR P42345 2/20 0.38
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
HPGD P15428 1/20 0.38
KMT2A Q03164 1/20 0.38
NAMPT P43490 4/20 0.37
RAB9A P51151 1/20 0.37
PTPN7 P35236 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8091717 0.91 CA2 (0.40) CA1CA2CA12CA4CA7
SCHEMBL8090705 0.89 NAMPT (0.40) CA1CA2CA12CA4CA7
SCHEMBL8104823 0.88 CA2 (0.39) CA1CA2CA12CA4CA7
SCHEMBL8091710 0.88 PIK3CD (0.36) CA1CA2CA12CA4CA7
SCHEMBL8091538 0.87 PIK3CD (0.43) PIK3CDPIK3CAMTOR
SCHEMBL8097257 0.87 ALDH1A1 (0.41) CA1CA2CA12CA4CA7
SCHEMBL8084009 0.87 PIK3CD (0.42) PIK3CDPIK3CAMTOR
SCHEMBL8104327 0.86 NAMPT (0.39) CA1CA2CA12CA4CA7
SCHEMBL8099408 0.86 CA2 (0.42) CA1CA2CA12CA4CA7
SCHEMBL8091534 0.86 NAMPT (0.40) ALDH1A1PIK3CDPIK3CAMTORMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed