SCHEMBL8105071

SCHEMBL8105071

CC(C)N(CCC1C(=O)CC1(C(=O)O)c1ccccc1)C(C)C

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 3/20 0.42
SIGMAR1 Q99720 1/20 0.38
SLC6A3 Q01959 3/20 0.37
SLC6A4 P31645 2/20 0.37
CYP2D6 P10635 1/20 0.37
HTR2C P28335 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4661013 0.76 SLC6A2 (0.44) SLC6A2SIGMAR1SLC6A3SLC6A4CYP2D6
Hydrochloric Acid SCHEMBL4021178 0.75 SLC6A2 (0.43) SLC6A2SIGMAR1SLC6A3SLC6A4CYP2D6
SCHEMBL8112597 0.75 SLC6A2 (0.43) SLC6A2SIGMAR1SLC6A3SLC6A4CYP2D6
SCHEMBL27499030 0.66 SLC22A1 (0.47) SLC6A2SLC6A4
SCHEMBL8105073 0.65 PRCP (0.53) SIGMAR1SLC6A4CYP2D6
Hydrochloric Acid SCHEMBL8320850 0.64 ALDH1A1 (0.51) SIGMAR1CYP2D6
Hydrochloric Acid SCHEMBL8107104 0.64 ALDH1A1 (0.54) SIGMAR1SLC6A4CYP2D6
Hydrochloric Acid SCHEMBL8097372 0.64 CHRM2 (0.45) SLC6A2SIGMAR1SLC6A4CYP2D6
Hydrochloric Acid SCHEMBL8106991 0.64 SLC6A2 (0.50) SLC6A2SIGMAR1SLC6A3SLC6A4CYP2D6
Hydrochloric Acid SCHEMBL8107066 0.64 CHRM2 (0.45) SLC6A2SIGMAR1SLC6A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6124354-A TREATMENT OF URINARY INCONTINENCE OR IRRITABLE BOWEL SYNDROME PHARMACIA & UPJOHN AB (SE) 2000-09-26 US disclosed
EP-0923536-A1 ARYLCYCLOALKANE CARBOXYLIC ESTERS, THEIR USE, PHARMACEUTICAL COMPOSITIONS AND PREPARATION Pharmacia & Upjohn Aktiebolag (SE) 1999-06-23 EP disclosed
WO-1998004517-A1 ARYLCYCLOALKANE CARBOXYLIC ESTERS, THEIR USE, PHARMACEUTICAL COMPOSITIONS AND PREPARATION PHARMACIA & UPJOHN AB (SE) 1998-02-05 WO disclosed