SCHEMBL8105481

SCHEMBL8105481

O=c1[nH]ccn1-c1ccc(OCC(F)(F)C(F)F)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.39
KMT2A Q03164 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CMA1 P23946 2/20 0.36
ACACB O00763 1/20 0.36
MMP13 P45452 1/20 0.36
MMP14 P50281 1/20 0.36
USP2 O75604 1/20 0.34
MAPT P10636 1/20 0.34
TSHR P16473 1/20 0.34
CYP2D6 P10635 1/20 0.31
SLC9A3 P48764 1/20 0.31
MEN1 O00255 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
CCNA2 P20248 1/20 0.30
CDK2 P24941 1/20 0.30
CCNA1 P78396 1/20 0.30
KCNH2 Q12809 1/20 0.30
MCHR1 Q99705 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8718847 0.93 ACACB (0.41) HTTKMT2ASMN1; SMN2ALDH1A1CMA1
SCHEMBL9016101 0.87 CMA1 (0.35) CMA1CYP2D6SLC9A3KCNH2MCHR1
SCHEMBL8723280 0.86 CMA1 (0.41) CMA1KCNH2MCHR1
SCHEMBL8723274 0.85 USP2 (0.46) SMN1; SMN2CMA1USP2MAPTTSHR
SCHEMBL8718863 0.84 CMA1 (0.37) ALDH1A1CMA1MMP13MMP14USP2
SCHEMBL8111166 0.81 TRPV1 (0.37) HTTALDH1A1CMA1MMP13MMP14
SCHEMBL6174527 0.79 HTT (0.46) HTTKMT2ASMN1; SMN2ALDH1A1CMA1
SCHEMBL7678488 0.77 HTT (0.41) HTTKMT2ASMN1; SMN2ALDH1A1CMA1
SCHEMBL7687627 0.76 HTT (0.39) HTTKMT2ASMN1; SMN2ALDH1A1ACACB
SCHEMBL8721198 0.76 POLB (0.49) KMT2ACMA1MAPTCYP2D6MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1033367-A2 Process for the preparation of optically active triazole derivatives and their imidazolidin-2-one intermediates TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-09-06 EP disclosed
US-5814324-A OIL IN WATER EMULSION COMPRISING ANTIFUNGAL TRIAZOLE COMPOUND DISPERSED IN WATER WITH FATTY ACID TRIGLYCERIDE, LECITHIN EMULSIFIER TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-09-29 US disclosed
US-5677464-A Production of optically active triazole compounds and their intermediates TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-10-14 US disclosed
EP-0746318-A1 INJECTABLE EMULSIONS CONTAINING ANTIFUNGAL TRIAZOLE DERIVATIVES Takeda Chemical Industries, Ltd. (JP) 1996-12-11 EP disclosed
EP-0687672-A2 Production of optically active triazole compounds and their intermediates TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-12-20 EP disclosed
WO-1995022973-A1 INJECTABLE EMULSIONS CONTAINING ANTIFUNGAL TRIAZOLE DERIVATIVES TAKEDA CHEMICALS INDUSTRIES, LTD. (JP) 1995-08-31 WO disclosed