SCHEMBL8106523

SCHEMBL8106523

Cc1ccc(-c2ccc(Cc3ncc(Cc4ccc(C#N)cc4)[nH]3)cc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRS3 P32247 6/20 0.54
HRH3 Q9Y5N1 3/20 0.47
CYP11B1 P15538 1/20 0.45
CYP11B2 P19099 1/20 0.45
ALDH1A1 P00352 2/20 0.43
CYP2A6 P11509 1/20 0.43
TSHR P16473 1/20 0.41
HSD17B10 Q99714 1/20 0.41
SCN10A Q9Y5Y9 1/20 0.41
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
CYP1A2 P05177 1/20 0.39
MAPT P10636 1/20 0.39
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39
CYP2C19 P33261 1/20 0.39
RECQL P46063 1/20 0.39
KMT2A Q03164 1/20 0.39
LOXL2 Q9Y4K0 1/20 0.38
KDM1A O60341 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7919393 0.89 BRS3 (0.62) BRS3HRH3CYP11B1CYP11B2CYP19A1
Hydrochloric Acid SCHEMBL8521500 0.88 BRS3 (0.61) BRS3HRH3CYP11B1CYP11B2CYP19A1
SCHEMBL8105207 0.88 BRS3 (0.53) BRS3HRH3CYP11B1CYP11B2TSHR
SCHEMBL8107069 0.88 BRS3 (0.51) BRS3HRH3CYP11B1CYP11B2ALDH1A1
SCHEMBL8106516 0.85 KIF11 (0.54) BRS3HRH3KDM1AMAOBCYP19A1
SCHEMBL8097328 0.84 BRS3 (0.49) BRS3HRH3ALDH1A1TSHRHSD17B10
SCHEMBL8306480 0.84 BRS3 (0.49) BRS3HRH3CYP11B1CYP11B2ALDH1A1
SCHEMBL8104996 0.84 BRS3 (0.62) BRS3HRH3CYP11B1CYP11B2
Hydrochloric Acid SCHEMBL8311538 0.84 KIF11 (0.52) BRS3HRH3KDM1AMAOBCYP19A1
SCHEMBL8498703 0.83 BRS3 (0.49) BRS3HRH3CYP11B1CYP11B2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0986302-A1 A METHOD OF TREATING CANCER Merck & Co., Inc. (US) 2000-03-22 EP disclosed
WO-1998054966-A1 A METHOD OF TREATING CANCER MERCK & CO., INC. (US) 1998-12-10 WO disclosed