SCHEMBL8306480

SCHEMBL8306480

N#Cc1ccc(Cc2cnc(Cc3ccc(-c4ccsc4)cc3)[nH]2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRS3 P32247 5/20 0.49
CYP17A1 P05093 1/20 0.44
CYP11B1 P15538 1/20 0.44
CYP11B2 P19099 1/20 0.44
LTA4H P09960 3/20 0.42
HRH3 Q9Y5N1 1/20 0.42
KDM1A O60341 1/20 0.40
ALDH1A1 P00352 2/20 0.38
SCN10A Q9Y5Y9 1/20 0.35
CYP2A6 P11509 2/20 0.35
TSHR P16473 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CYP2E1 P05181 1/20 0.34
CYP2B6 P20813 1/20 0.34
TYMP P19971 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
CYP1A2 P05177 1/20 0.34
MAPT P10636 1/20 0.34
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8310148 0.99 BRS3 (0.48) BRS3CYP17A1CYP11B1CYP11B2LTA4H
SCHEMBL8106523 0.84 BRS3 (0.54) BRS3CYP11B1CYP11B2HRH3KDM1A
SCHEMBL7919393 0.84 BRS3 (0.62) BRS3CYP11B1CYP11B2HRH3
Hydrochloric Acid SCHEMBL8521500 0.83 BRS3 (0.61) BRS3CYP11B1CYP11B2HRH3
SCHEMBL8105207 0.83 BRS3 (0.53) BRS3CYP11B1CYP11B2HRH3SCN10A
SCHEMBL8106516 0.80 KIF11 (0.54) BRS3HRH3KDM1A
Hydrochloric Acid SCHEMBL8311538 0.79 KIF11 (0.52) BRS3HRH3KDM1A
SCHEMBL8498703 0.78 BRS3 (0.49) BRS3CYP11B1CYP11B2HRH3ALDH1A1
SCHEMBL8107069 0.78 BRS3 (0.51) BRS3CYP11B1CYP11B2HRH3KDM1A
SCHEMBL8097365 0.77 BRS3 (0.50) BRS3HRH3TSHRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0891343-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 1999-01-20 EP claimed
WO-1997036886-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 1997-10-09 WO claimed