SCHEMBL8106631

SCHEMBL8106631

C[C@H](CO)NC(=O)Nc1ccc(-c2nc(NCCO)cc(C3(S(=O)(=O)CCCO)CCC3)n2)cc1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.35
GPR119 Q8TDV5 1/20 0.35
PIK3CD O00329 7/20 0.34
PIK3CA P42336 6/20 0.34
MTOR P42345 3/20 0.34
PIK3CB P42338 1/20 0.34
PIK3CG P48736 1/20 0.34
PDGFRB P09619 2/20 0.32
KDR P35968 2/20 0.32
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32
P2RY12 Q9H244 1/20 0.30
RAF1 P04049 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8106629 0.85 PIK3CD (0.34) CYP1A2GPR119PIK3CDPIK3CAMTOR
SCHEMBL8100159 0.85 PIK3CA (0.36) CYP1A2GPR119PIK3CDPIK3CAMTOR
SCHEMBL8098280 0.83 RAB9A (0.39) CYP1A2GPR119PIK3CDPIK3CAMTOR
SCHEMBL8091770 0.82 MTOR (0.37) CYP1A2GPR119PIK3CDPIK3CAMTOR
SCHEMBL8091937 0.80 CA12 (0.39) PIK3CDPIK3CAMTORCA12CA1
SCHEMBL3924188 0.79 PIK3CA (0.56) PIK3CDPIK3CAMTORPIK3CBPIK3CG
SCHEMBL3935410 0.79 PIK3CA (0.56) PIK3CDPIK3CAMTORPIK3CBPIK3CG
SCHEMBL8098837 0.79 PIK3CA (0.40) PIK3CDPIK3CAMTORPIK3CBPIK3CG
SCHEMBL8100894 0.78 PIK3CD (0.37) CYP1A2GPR119PIK3CDPIK3CAMTOR
SCHEMBL8091352 0.77 PIK3CA (0.41) PIK3CDPIK3CAMTORPIK3CBPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed