SCHEMBL8106919

SCHEMBL8106919

C=C(C)COc1c(Br)cc(Br)cc1C(C)C

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.42
GABRB1 P18505 1/20 0.42
THRB P10828 7/20 0.32
THRA P10827 6/20 0.32
HSD17B10 Q99714 1/20 0.32
RXRA P19793 1/20 0.32
LMNA P02545 2/20 0.32
SRD5A2 P31213 1/20 0.32
AKR1B1 P15121 1/20 0.32
ALOX15 P16050 1/20 0.31
ALOX12 P18054 1/20 0.31
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
MAPT P10636 1/20 0.30
MAPK1 P28482 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9181295 0.85 HSD17B10 (0.38) THRBTHRAHSD17B10LMNAAKR1B1
SCHEMBL28891144 0.80 GABRA1 (0.42) GABRA1GABRB1THRBTHRAHSD17B10
SCHEMBL670896 0.79 MEN1 (0.44) HSD17B10LMNAAKR1B1ALOX15ALOX12
SCHEMBL7062178 0.76 TSHR (0.40) GABRA1GABRB1THRBTHRAHSD17B10
SCHEMBL15709517 0.75 PTGDR2 (0.39) HSD17B10LMNAAKR1B1ALOX15ALOX12
SCHEMBL7067884 0.75 THRB (0.40) GABRA1GABRB1THRBTHRAHSD17B10
SCHEMBL1805856 0.74 TSHR (0.44) GABRA1GABRB1THRBTHRAMEN1
SCHEMBL7618929 0.74 GABRA1 (0.41) GABRA1GABRB1THRBTHRAHSD17B10
SCHEMBL1535013 0.74 GABRA1 (0.37) GABRA1GABRB1THRBTHRALMNA
SCHEMBL4646137 0.74 GABRA1 (0.41) GABRA1GABRB1THRBTHRALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6093838-A FOR TREATING SKIN-RELATED DISEASES, INCLUDING ACTINIC KERATOSES, ARSENIC KERATOSES, ECZEMA ALLERGAN SALES, INC. (US) 2000-07-25 US disclosed