SCHEMBL8107629

SCHEMBL8107629

COc1ccc(CN2CCC(=O)CC2)cc1.COc1ccc(CN2CCC(=O)CC2)cc1

nearest known ligand 0.67

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.65
SMN1; SMN2 Q16637 1/20 0.63
GAA P10253 1/20 0.59
PTGIR P43119 1/20 0.58
TACR1 P25103 1/20 0.57
HRH3 Q9Y5N1 2/20 0.57
CMA1 P23946 1/20 0.56
CHKA P35790 1/20 0.54
POLB P06746 1/20 0.54
PKM P14618 1/20 0.54
GSK3A P49840 1/20 0.53
GSK3B P49841 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1586605 1.00 SIGMAR1 (0.65) SIGMAR1SMN1; SMN2GAAPTGIRTACR1
SCHEMBL3979749 0.94 PTGIR (0.60) SIGMAR1SMN1; SMN2GAAPTGIRTACR1
SCHEMBL9829472 0.90 ABCB1 (0.57) SIGMAR1SMN1; SMN2GAAPTGIRTACR1
SCHEMBL20804352 0.85 SIGMAR1 (0.85) SIGMAR1SMN1; SMN2PTGIRCHKAPOLB
SCHEMBL1043952 0.85 SIGMAR1 (0.85) SIGMAR1SMN1; SMN2PTGIRCHKAPOLB
SCHEMBL19285228 0.85 SIGMAR1 (0.85) SIGMAR1SMN1; SMN2PTGIRCHKAPOLB
SCHEMBL3714297 0.83 SIGMAR1 (0.75) SIGMAR1HRH3GSK3AGSK3B
SCHEMBL12403963 0.83 KMT2A (0.51) SIGMAR1TACR1HRH3
SCHEMBL3171551 0.82 PTGIR (0.81) SIGMAR1SMN1; SMN2PTGIRHRH3CHKA
SCHEMBL28048490 0.82 PTGIR (0.75) SIGMAR1SMN1; SMN2PTGIRHRH3CHKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1056744-A1 6,9-DISUBSTITUTED 2- TRANS-(4- AMINOCYCLOHEXYL) AMINO]PURINES Aventis Pharmaceuticals Inc. (US) 2000-12-06 EP disclosed
WO-1999043675-A1 6,9-DISUBSTITUTED 2-[TRANS-(4- AMINOCYCLOHEXYL) AMINO]PURINES AVENTIS PHARMACEUTICALS INC. (US) 1999-09-02 WO disclosed