SCHEMBL8107664

SCHEMBL8107664

CN1C2CCC1CC(c1cncc3ccccc13)C2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.39
SLC6A3 Q01959 2/20 0.39
CNR1 P21554 1/20 0.38
CNR2 P34972 1/20 0.38
DRD2 P14416 3/20 0.37
CHRM3 P20309 2/20 0.37
SLC6A4 P31645 2/20 0.37
DRD3 P35462 2/20 0.37
CHRM2 P08172 1/20 0.37
CHRM4 P08173 1/20 0.37
CHRM5 P08912 1/20 0.37
ADRA2A P08913 1/20 0.37
CHRM1 P11229 1/20 0.37
ADRA2B P18089 1/20 0.37
ADRA2C P18825 1/20 0.37
DRD1 P21728 1/20 0.37
HRH2 P25021 1/20 0.37
ADRA1D P25100 1/20 0.37
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1177800 0.83 ROCK2 (0.42) CNR1CNR2DRD2SLC6A4CYP3A4
SCHEMBL1177802 0.83 ROCK2 (0.42) CNR1CNR2DRD2SLC6A4CYP3A4
SCHEMBL13728399 0.79 CYP11B2 (0.42) CNR1CNR2DRD2SLC6A4ADRA2A
Bromide SCHEMBL8108934 0.77 HRH3 (0.37) CYP11B2
SCHEMBL28442398 0.76 TDP1 (0.41) CNR1CNR2DRD2SLC6A4ADRA2A
Cyclohexane SCHEMBL22288135 0.74 TDP1 (0.44) CNR1CNR2ADRA2AADRA2BADRA2C
SCHEMBL11665783 0.74 TDP1 (0.44) CNR1CNR2ADRA2AADRA2BADRA2C
Fumaric Acid SCHEMBL1177870 0.74 KDM4E (0.41)
SCHEMBL30735834 0.72 HTR2C (0.49) SLC6A2SLC6A3SLC6A4HTR2CHTR6
SCHEMBL7963921 0.72 HTR2C (0.49) SLC6A2SLC6A3SLC6A4HTR2CHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6107307-A PSYCHOLOGICAL DISORDERS ELI LILLY AND COMPANY (US) 2000-08-22 US disclosed
EP-0969005-A1 Azabicyclic inhibitors of serotonin reuptake ELI LILLY AND COMPANY (US) 2000-01-05 EP disclosed